Council Regulation (EC) No 129/2007 of 12 February 2007 providing for duty-free t... (32007R0129)
EU - Rechtsakte: 02 Customs Union and free movement of goods

COUNCIL REGULATION (EC) No 129/2007

of 12 February 2007

providing for duty-free treatment for specified pharmaceutical active ingredients bearing an ‘international non-proprietary name’ (INN) from the World Health Organisation and specified products used for the manufacture of finished pharmaceuticals and amending Annex I to Regulation (EEC) No 2658/87

THE COUNCIL OF THE EUROPEAN UNION,
Having regard to the Treaty establishing the European Community, and in particular Article 133 thereof,
Having regard to the proposal from the Commission,
Whereas:
(1) In the course of the Uruguay Round negotiations, the Community and a number of countries agreed that duty-free treatment should be granted to pharmaceutical products falling within the Harmonised System (HS) Chapter 30 and HS headings 2936, 2937, 2939 and 2941 as well as to designated pharmaceutical active ingredients bearing an ‘international non-proprietary name’ (INN) from the World Health Organisation, specified salts, esters or hydrates of such INNs, and designated intermediates used for the production and manufacture of finished products.
(2) The results of the discussions, as set out in the record of discussions, were incorporated into the tariff schedules of the participants, annexed to the Marrakesh Protocol to the GATT 1994.
(3) Participants concluded that representatives of the WTO members, party to the record of discussions, would meet under the auspices of the WTO Council for Trade in Goods, normally at least once every three years to review the product coverage with a view to including, by consensus, additional pharmaceutical products for tariff elimination.
(4) In the course of three such reviews it was concluded that a certain number of additional INNs and intermediates used for production and manufacture of finished pharmaceuticals should be granted duty-free treatment, that certain of these intermediates should be transferred to the list of INNs, and that the list of specified prefixes and suffixes for salts, esters or hydrates of INNs should be expanded.
(5) Council Regulation (EEC) No 2658/87 of 23 July 1987 on the tariff and statistical nomenclature and on the Common Customs Tariff (1) established the Combined Nomenclature (CN) and set out the conventional duty rates of the Common Customs Tariff.
(6) Regulation (EEC) No 2658/87 should therefore be amended accordingly,
HAS ADOPTED THIS REGULATION:

Article 1

As from 1 January 2007 the Community shall extend duty-free treatment to the INNs listed in Annex I.

Article 2

As from 1 January 2007 the list of prefixes and suffixes which, in combination with the INNs, describe the salts, esters or hydrates of INNs which are also eligible for duty-free treatment, on condition that they are classifiable in the same six-digit HS-subheading as the corresponding INN, shall be replaced by the list in Annex II.

Article 3

As from 1 January 2007 the Community shall extend duty-free treatment to the intermediates used in the production and manufacture of pharmaceutical products listed in Annex III.

Article 4

As from 1 January 2007 the intermediates listed in Annex IV shall no longer benefit from duty-free treatment.

Article 5

Annexes 3, 4 and 6 of Section II of Part three of Annex I to Regulation (EEC) No 2658/87 (Lists of pharmaceutical substances which qualify for duty-free treatment) shall be amended accordingly.

Article 6

This Regulation shall enter into force on the day following its publication in the
Official Journal of the European Union
.
This Regulation shall be binding in its entirety and directly applicable in all Member States.
Done at Brussels, 12 February 2007.
For the Council
The President
F.-W. STEINMEIER
(1)  
OJ L 256, 7.9.1987, p. 1
. Regulation as last amended by Regulation (EC) No 1930/2006 (
OJ L 406, 30.12.2006, p. 9
).

ANNEX I

List of international non-proprietary names (INNs) to be added to the list of products receiving duty-free treatment included in Annex 3 to Commission Regulation (EC) No 1549/2006 (1)

ID No

CN code

CAS RN

Name

696

2842 90 80

12539-23-0

vangatalcite

572

2843 90 90

129580-63-8

satraplatin

413

2843 90 90

141977-79-9

miriplatin

223

2843 90 90

146665-77-2

eptaplatin

682

2843 90 90

172903-00-3

triplatin tetranitrate

504

2843 90 90

181630-15-9

picoplatin

807

2843 90 90

274679-00-4

padoporfin

629

2844 40 30

131608-78-1

technetium (99mTc) nitridocade

628

2844 40 30

225239-31-6

technetium (99mTc) fanolesomab

711

2844 40 30

476413-07-7

yttrium (90Y) tacatuzumab tetraxetan (yttrium (90Y) tacatuzumab)

738

2845 90 10

474641-19-5

deutolperisone

283

2846 90 00

193901-90-5

gadofosveset

284

2846 90 00

227622-74-4

gadomelitol

281

2846 90 00

280776-87-6

gadocoletic acid

282

2846 90 00

544697-52-1

gadodenterate

761

2903 39 90

354-92-7

perflisobutane

497

2903 39 90

355-25-9

perflubutane

495

2903 39 90

355-42-0

perflexane

498

2903 39 90

76-19-7

perflutren

496

2903 47 00

307-43-7

perflubrodec

328

2906 19 00

163217-09-2

inecalcitol

727

2906 19 00

524067-21-8

becocalcidiol

21

2907 29 00

57-91-0

alfatradiol

464

2909 49 90

128607-22-7

ospemifene

66

2909 49 90

302904-82-1

atocalcitol

270

2909 49 90

341524-89-8

fispemifene

592

2909 50 90

3380-30-1

soneclosan

335

2914 40 90

158440-71-2

irofulven

803

2914 70 00

274925-86-9

nebicapone

56

2915 90 80

185517-21-9

arundic acid

87

2916 39 00

153559-49-0

bexarotene

640

2918 19 85

121009-77-6

tenivastatin

659

2918 19 85

156965-06-9

tisocalcitate

750

2918 19 85

54845-95-3

icomucret

677

2918 99 90

157283-68-6

travoprost

744

2918 99 90

161172-51-6

etalocib

294

2918 99 90

183293-82-5

gemcabene

643

2918 99 90

251565-85-2

tesaglitazar

757

2918 99 90

476436-68-7

naveglitazar

436

2921 30 99

219810-59-0

neramexane

153

2921 49 80

186495-49-8

delucemine

124

2921 49 80

226256-56-0

cinacalcet

367

2921 49 80

33817-09-3

levmetamfetamine

234

2922 19 80

119618-22-3

esoxybutynin

611

2922 19 80

146376-58-1

talibegron

596

2922 19 80

148717-90-2

squalamine

266

2922 19 80

162359-55-9

fingolimod

683

2922 19 80

186139-09-3

trodusquemine

193

2922 19 80

190258-12-9

edronocaine

709

2922 19 80

207916-33-4

xidecaflur

391

2922 19 80

36144-08-8

mantabegron

644

2922 19 80

98774-23-3

tesmilifene

626

2922 29 00

148717-54-8

tecalcet

619

2922 29 00

175591-23-8

tapentadol

440

2922 29 00

90060-42-7

nolomirole

230

2922 39 00

33643-46-8

esketamine

198

2922 49 95

176199-48-7

eglumetad (eglumegad)

310

2922 49 95

198022-65-0

icofungipen

386

2922 49 95

220991-20-8

lumiracoxib

554

2922 49 95

220991-32-2

robenacoxib

103

2922 50 00

135306-78-4

caloxetic acid

72

2922 50 00

187219-95-0

axomadol

278

2922 50 00

193901-91-6

fosveset

589

2922 50 00

252920-94-8

solabegron

551

2922 50 00

255734-04-4

ritobegron

752

2922 50 00

269079-62-1

isalmadol

261

2922 50 00

286930-03-8

fesoterodine

238

2922 50 00

37178-37-3

etilevodopa

399

2922 50 00

7101-51-1

melevodopa

161

2922 50 00

93413-62-8

desvenlafaxine

110

2924 19 00

1188-38-1

carglumic acid

632

2924 19 00

250694-07-6

teglicar

692

2924 19 00

92262-58-3

valrocemide

603

2924 29 95

112522-64-2

tacedinaline

36

2924 29 95

119363-62-1

amiglumide

195

2924 29 95

131179-95-8

efaproxiral

528

2924 29 95

133865-88-0

ralfinamide

567

2924 29 95

133865-89-1

safinamide

735

2924 29 95

147497-64-1

davasaicin

71

2924 29 95

156740-57-7

axitirome

434

2924 29 95

163000-63-3

neboglamine (nebostinel)

26

2924 29 95

173334-57-1

aliskiren

347

2924 29 95

175481-36-4

lacosamide (erlosamide)

332

2924 29 95

181872-90-2

iosimenol

568

2924 29 95

183990-46-7

salcaprozic acid

279

2924 29 95

188196-22-7

frakefamide

601

2924 29 95

193079-69-5

tabimorelin

462

2924 29 95

196618-13-0

oseltamivir

349

2924 29 95

209394-27-4

ladostigil

828

2924 29 95

220847-86-9

valategrast

614

2924 29 95

228266-40-8

taltobulin

668

2924 29 95

260980-89-0

topilutamide

720

2924 29 95

387825-03-8

salclobuzic acid

772

2924 29 95

441765-98-6

talaglumetad

51

2924 29 95

67346-49-0

arformoterol

449

2925 29 00

146510-36-3

olanexidine

45

2925 29 00

170368-04-4

anisperimus

494

2925 29 00

229614-55-5

peramivir

737

2925 29 00

287096-87-1

delmitide

35

2925 29 00

346735-24-8

amelubant

642

2926 90 95

108605-62-5

teriflunomide

121

2926 90 95

153259-65-5

cilomilast

801

2926 90 95

202057-76-9

manitimus

428

2926 90 95

220641-11-2

naminidil

219

2928 00 90

130579-75-8

eplivanserin

570

2928 00 90

149400-88-4

sardomozide

777

2928 00 90

154039-60-8

marimastat

798

2928 00 90

203737-93-3

istaroxime

576

2928 00 90

352513-83-8

semapimod

398

2928 00 90

76144-81-5

meldonium

75

2929 90 00

136470-65-0

banoxantrone

69

2929 90 00

166518-60-1

avasimibe

172

2929 90 00

168021-79-2

disufenton sodium

833

2930 90 30

583-91-5

desmeninol

233

2930 90 85

101973-77-7

esonarimod

53

2930 90 85

112111-43-0

armodafinil

731

2930 90 85

158382-37-7

canfosfamide

618

2930 90 85

179545-77-8

tanomastat

766

2930 90 85

187870-78-6

rimeporide

196

2930 90 85

202340-45-2

eflucimibe

165

2930 90 85

29335-92-0

dextiopronin

760

2930 90 85

496050-39-6

pemaglitazar

250

2930 90 85

59973-80-7

exisulind

307

2931 00 95

133208-93-2

ibrolipim

372

2931 00 95

63132-38-7

lidadronic acid

556

2932 19 00

156722-18-8

rostafuroxin

410

2932 19 00

393101-41-2

milataxel

58

2932 29 85

109791-32-4

ascorbyl gamolenate

171

2932 29 85

127943-53-7

disermolide

272

2932 29 85

140616-46-2

fluorescein lisicol

19

2932 29 85

150785-53-8

alemcinal

416

2932 29 85

154738-42-8

mitemcinal

38

2932 29 85

161262-29-9

amotosalen

555

2932 29 85

162011-90-7

rofecoxib

574

2932 29 85

165108-07-6

selamectin

269

2932 29 85

189954-96-9

firocoxib

469

2932 99 50

186040-50-6

paclitaxel ceribate

273

2932 99 70

114870-03-0

fondaparinux sodium

229

2932 99 70

128196-01-0

escitalopram

463

2932 99 70

137275-81-1

osemozotan

312

2932 99 70

149920-56-9

idraparinux sodium

211

2932 99 70

167256-08-8

enrasentan

150

2932 99 70

171092-39-0

defoslimod

650

2932 99 70

175013-73-7

tidembersat

455

2932 99 70

181296-84-4

omigapil

743

2932 99 70

185955-34-4

eritoran

461

2932 99 70

186348-23-2

ortataxel

529

2932 99 70

196597-26-9

ramelteon

467

2932 99 70

280585-34-4

oxeglitazar

375

2932 99 70

329306-27-6

lirimilast

163

2932 99 70

51372-29-3

dexbudesonide

54

2932 99 70

75887-54-6

artemotil

314

2932 99 70

81267-65-4

idronoxil

667

2932 99 85

175013-84-0

tonabersat

109

2932 99 85

184653-84-7

carabersat

55

2932 99 85

81496-81-3

artenimol

769

2932 99 90

343306-71-8

sugammadex

224

2933 29 90

129805-33-0

eptotermin alfa

255

2933 29 90

134183-95-2

fampronil

249

2933 29 90

141758-74-9

exenatide

806

2933 29 90

144689-24-7

olmesartan

176

2933 29 90

149838-23-3

doranidazole

268

2933 29 90

150586-58-6

fipamezole

578

2933 29 90

154906-40-8

semparatide

204

2933 29 90

159075-60-2

emfilermin

209

2933 29 90

159519-65-0

enfuvirtide

472

2933 29 90

162394-19-6

palifermin

89

2933 29 90

163796-60-9

bifarcept

321

2933 29 90

170105-16-5

imidafenacin

657

2933 29 90

178823-49-9

tiplimotide

253

2933 29 90

189353-31-9

fadolmidine (radolmidine)

389

2933 29 90

200074-80-2

lusupultide

126

2933 29 90

213027-19-1

cipralisant

541

2933 29 90

219527-63-6

repifermin

605

2933 29 90

220712-29-8

tadekinig alfa

167

2933 29 90

246539-15-1

dibotermin alfa

536

2933 29 90

259188-38-0

rebimastat

790

2933 29 90

444069-80-1

dapiclermine

396

2933 29 90

478166-15-3

mecasermin rinfabate

134

2933 39 99

0-00-0

crobenetine

591

2933 39 99

0-00-0

solimastat

159

2933 39 99

100643-71-8

desloratadine

299

2933 39 99

103766-25-2

gimeracil

342

2933 39 99

112568-12-4

iturelix

637

2933 39 99

113712-98-4

tenatoprazole

232

2933 39 99

119141-88-7

esomeprazole

804

2933 39 99

119229-65-1

nerispirdine

308

2933 39 99

119515-38-7

icaridin

29

2933 39 99

120241-31-8

alvameline

411

2933 39 99

128420-61-1

minopafant

678

2933 39 99

134234-12-1

traxoprodil

519

2933 39 99

134457-28-6

prazarelix

791

2933 39 99

138530-94-6

dexlansoprazole

800

2933 39 99

138530-95-7

levolansoprazole

712

2933 39 99

142852-50-4

zanapezil

252

2933 39 99

147116-64-1

ezlopitant

394

2933 39 99

147116-67-4

maropitant

180

2933 39 99

150337-94-3

ecalcidene

350

2933 39 99

153322-05-5

lanicemine

815

2933 39 99

15585-43-0

rivanicline

30

2933 39 99

156053-89-3

alvimopan

333

2933 39 99

166181-63-1

ipravacaine

707

2933 39 99

168266-90-8

vofopitant

549

2933 39 99

168273-06-1

rimonabant

215

2933 39 99

170364-57-5

enzastaurin

318

2933 39 99

172152-36-2

ilaprazole

107

2933 39 99

178979-85-6

capravirine

655

2933 39 99

179033-51-3

timcodar

262

2933 39 99

183305-24-0

fidexaban

809

2933 39 99

188396-77-2

paliroden

158

2933 39 99

188913-58-8

dersalazine

125

2933 39 99

190648-49-8

cipemastat

465

2933 39 99

193153-04-7

otamixaban

380

2933 39 99

193275-84-2

lonafarnib

645

2933 39 99

195875-84-4

tesofensine

623

2933 39 99

198283-73-7

tebanicline

507

2933 39 99

198480-55-6

pipendoxifene

65

2933 39 99

198904-31-3

atazanavir

199

2933 39 99

198958-88-2

elarofiban

341

2933 39 99

201605-51-8

itriglumide

91

2933 39 99

202189-78-4

bilastine

240

2933 39 99

202409-33-4

etoricoxib

649

2933 39 99

202590-69-0

ticalopride

325

2933 39 99

204205-90-3

indibulin

136

2933 39 99

211914-51-1

dabigatran

137

2933 39 99

211915-06-9

dabigatran etexilate

701

2933 39 99

212141-54-3

vatalanib

74

2933 39 99

215529-47-8

bamirastine

10

2933 39 99

227940-00-3

adekalant

699

2933 39 99

249296-44-4

varenicline

797

2933 39 99

252870-53-4

ispronicline

76

2933 39 99

263562-28-3

barixibat

594

2933 39 99

284461-73-0

sorafenib

821

2933 39 99

288104-79-0

surinabant

52

2933 39 99

289893-25-0

arimoclomol

721

2933 39 99

370893-06-4

ancriviroc

392

2933 39 99

376348-65-1

maraviroc

164

2933 39 99

40431-64-9

dexmethylphenidate

316

2933 39 99

58754-46-4

iferanserin

788

2933 39 99

64881-21-6

caricotamide

409

2933 39 99

72599-27-0

miglustat

627

2933 39 99

75970-99-9

tecastemizole

579

2933 39 99

98326-32-0

senazodan

448

2933 49 10

167887-97-0

olamufloxacin

606

2933 49 90

106635-80-7

tafenoquine

714

2933 49 90

139233-53-7

zelandopam

25

2933 49 90

144506-11-6

alilusem

397

2933 49 90

146362-70-1

meclinertant (reminertant)

508

2933 49 90

147511-69-1

pitavastatin (itavastatin)

506

2933 49 90

149759-26-2

pinokalant

613

2933 49 90

174636-32-9

talnetant

290

2933 49 90

194804-75-6

garenoxacin

515

2933 49 90

195532-12-8

pradofloxacin

352

2933 49 90

197509-46-9

laniquidar

622

2933 49 90

206873-63-4

tariquidar

288

2933 49 90

213998-46-0

gantacurium chloride

717

2933 49 90

241800-98-6

zoniporide

590

2933 49 90

242478-37-1

solifenacin

492

2933 49 90

257933-82-7

pelitinib

672

2933 49 90

262352-17-0

torcetrapib

476

2933 49 90

540769-28-6

palosuran

586

2933 49 90

57695-04-2

sitamaquine

264

2933 59 95

0-00-0

figopitant

660

2933 59 95

103024-93-7

tiviciclovir

406

2933 59 95

117414-74-1

midafotel

452

2933 59 95

124265-89-0

omaciclovir

173

2933 59 95

129716-58-1

dofequidar

102

2933 59 95

133804-44-1

caldaret

366

2933 59 95

138117-50-7

leteprinim

213

2933 59 95

142217-69-4

entecavir

763

2933 59 95

146464-95-1

pralatrexate

641

2933 59 95

147127-20-6

tenofovir

531

2933 59 95

147254-64-6

ranirestat

205

2933 59 95

149950-60-7

emivirine

320

2933 59 95

152459-95-5

imatinib

511

2933 59 95

153537-73-6

plevitrexed

100

2933 59 95

153808-85-6

cadrofloxacin

503

2933 59 95

154889-68-6

pibrozelesin

718

2933 59 95

167354-41-8

zosuquidar

174

2933 59 95

170912-52-4

donitriptan

146

2933 59 95

171714-84-4

darusentan

32

2933 59 95

177036-94-1

ambrisentan

226

2933 59 95

183321-74-6

erlotinib

768

2933 59 95

186692-46-6

seliciclib

17

2933 59 95

187949-02-6

albaconazole

381

2933 59 95

192725-17-0

lopinavir

16

2933 59 95

193681-12-8

alamifovir

691

2933 59 95

195157-34-7

valomaciclovir

254

2933 59 95

196612-93-8

falnidamol

547

2933 59 95

199463-33-7

revaprazan

260

2933 59 95

204267-33-4

feloprentan

450

2933 59 95

204697-65-4

olcegepant

746

2933 59 95

209799-67-7

forodesine

716

2933 59 95

210245-80-0

zonampanel

162

2933 59 95

220984-26-9

detiviciclovir

142

2933 59 95

244767-67-7

dapivirine

208

2933 59 95

259525-01-4

enecadin

241

2933 59 95

269055-15-4

etravirine

439

2933 59 95

290297-26-6

netupitant

566

2933 59 95

324758-66-9

sabiporide

724

2933 59 95

330784-47-9

avanafil

703

2933 59 95

334476-46-9

vestipitant

753

2933 59 95

336113-53-2

ispinesib

695

2933 59 95

338992-00-0

vandetanib

725

2933 59 95

354813-19-7

balicatib

616

2933 59 95

387867-13-2

tandutinib

242

2933 59 95

402595-29-3

etriciguat

522

2933 59 95

443144-26-1

pruvanserin

548

2933 59 95

500287-72-9

rilpivirine

147

2933 59 95

569351-91-3

dasantafil

795

2933 59 95

61337-87-9

esmirtazapine

222

2933 69 80

179756-85-5

eptapirone

728

2933 69 80

187393-00-6

bemotrizinol

512

2933 69 80

69004-04-2

ponazuril

466

2933 69 80

937-13-3

oteracil

235

2933 79 00

138729-47-2

eszopiclone

354

2933 79 00

142139-60-4

lapisteride

111

2933 79 00

147568-66-9

carmoterol

88

2933 79 00

148905-78-6

bexlosteride

296

2933 79 00

160135-92-2

gemopatrilat

156

2933 79 00

161982-62-3

depreotide

251

2933 79 00

163222-33-1

ezetimibe

140

2933 79 00

182821-27-8

daglutril

271

2933 79 00

187523-35-9

flindokalner

120

2933 79 00

188968-51-6

cilengitide

362

2933 79 00

191732-72-6

lenalidomide

656

2933 79 00

192185-72-1

tipifarnib

577

2933 79 00

194413-58-6

semaxanib

355

2933 79 00

248281-84-7

laquinimod

823

2933 79 00

254964-60-8

tasquinimod

324

2933 79 00

312753-06-3

indacaterol

787

2933 79 00

357336-20-0

brivaracetam

818

2933 79 00

357336-74-4

seletracetam

781

2933 79 00

503612-47-3

apixaban

820

2933 79 00

557795-19-4

sunitinib

231

2933 99 30

104746-04-5

eslicarbazepine

181

2933 99 30

112108-01-7

ecopipam

422

2933 99 30

137975-06-5

mozavaptan

665

2933 99 30

150683-30-0

tolvaptan

131

2933 99 30

210101-16-9

conivaptan

370

2933 99 30

29331-92-8

licarbazepine

500

2933 99 40

144912-63-0

perzinfotel

378

2933 99 40

168079-32-1

lixivaptan

423

2933 99 40

174391-92-5

mozenavir

166

2933 99 40

82059-50-5

dextofisopam

730

2933 99 90

103597-45-1

bisoctrizole

597

2933 99 90

106344-20-1

stannsoporfin

811

2933 99 90

110078-46-1

plerixafor

610

2933 99 90

110230-98-3

talaporfin

46

2933 99 90

114560-48-4

apaziquone

778

2933 99 90

129497-78-5

verteporfin

510

2933 99 90

144510-96-3

pixantrone

544

2933 99 90

144875-48-9

resiquimod

631

2933 99 90

145158-71-0

tegaserod

588

2933 99 90

149606-27-9

soblidotin

770

2933 99 90

149682-77-9

talabostat

101

2933 99 90

151878-23-8

calcobutrol

518

2933 99 90

153804-05-8

pratosartan

758

2933 99 90

154082-13-0

omocianine

442

2933 99 90

156090-17-4

nortopixantrone

669

2933 99 90

156090-18-5

topixantrone

371

2933 99 90

156897-06-2

licofelone

267

2933 99 90

160146-17-8

finrozole

582

2933 99 90

160970-54-7

silodosin

311

2933 99 90

169543-49-1

icrocaptide

700

2933 99 90

172732-68-2

varespladib

435

2933 99 90

173240-15-8

nemifitide

210

2933 99 90

176644-21-6

eniporide

323

2933 99 90

177469-96-4

implitapide

457

2933 99 90

178040-94-3

opaviraline

28

2933 99 90

179120-92-4

altinicline

97

2933 99 90

179324-69-7

bortezomib

600

2933 99 90

179386-43-7

sumanirole

357

2933 99 90

180916-16-9

lasofoxifene

64

2933 99 90

182316-31-0

ataquimast

329

2933 99 90

186392-65-4

ingliforib

80

2933 99 90

188696-80-2

becampanel

471

2933 99 90

189198-30-9

pactimibe

421

2933 99 90

189752-49-6

motexafin

822

2933 99 90

192658-64-3

tasidotin

710

2933 99 90

192939-46-1

ximelagatran

108

2933 99 90

193273-66-4

capromorelin

276

2933 99 90

194798-83-9

fosfluconazole

79

2933 99 90

198481-32-2

bazedoxifene

149

2933 99 90

201530-41-8

deferasirox

98

2933 99 90

203258-60-0

brostallicin

454

2933 99 90

204248-78-2

omiganan

295

2933 99 90

204519-64-2

gemifloxacin

523

2933 99 90

207993-12-2

pumafentrine

361

2933 99 90

215808-49-4

lemuteporfin

826

2933 99 90

21919-05-1

tretazicar

831

2933 99 90

219680-11-2

zabofloxacin

526

2933 99 90

244081-42-3

rafabegron

755

2933 99 90

248919-64-4

linaprazan

652

2933 99 90

251562-00-2

tifuvirtide

595

2933 99 90

261944-46-1

soraprazan

705

2933 99 90

274901-16-5

vildagliptin

557

2933 99 90

284041-10-7

rostaporfin

767

2933 99 90

361442-04-8

saxagliptin

447

2933 99 90

38101-59-6

oglufanide

133

2933 99 90

38609-97-1

cridanimod

481

2933 99 90

396091-73-9

pasireotide

139

2933 99 90

404951-53-7

dacinostat

192

2933 99 90

433922-67-9

edratide

170

2933 99 90

481658-94-0

dirlotapide

723

2933 99 90

533927-56-9

atilmotin

773

2933 99 90

637328-69-9

tanogitran

681

2933 99 90

72741-87-8

tridolgosir

754

2933 99 90

82059-51-6

levotofisopam

419

2934 10 00

130112-42-4

mivotilate

144

2934 10 00

139226-28-1

darbufelone

259

2934 10 00

144060-53-7

febuxostat

646

2934 10 00

145739-56-6

tetomilast

438

2934 10 00

161600-01-7

netoglitazone

534

2934 10 00

182760-06-1

ravuconazole

6

2934 10 00

185106-16-5

acotiamide

553

2934 10 00

185428-18-6

rivoglitazone

73

2934 10 00

199113-98-9

balaglitazone

186

2934 10 00

213411-83-7

edaglitazone

736

2934 10 00

239101-33-8

deferitrin

122

2934 10 00

300832-84-2

ciluprevir

15

2934 10 00

341028-37-3

alagebrium chloride

819

2934 10 00

342026-92-0

sipoglitazar

550

2934 10 00

79714-31-1

risarestat

580

2934 20 80

154189-40-9

sibenadet

344

2934 20 80

176975-26-1

izonsteride

373

2934 20 80

245116-90-9

lidorestat

387

2934 20 80

367514-87-2

lurasidone

105

2934 99 90

0-00-0

cangrelor

287

2934 99 90

0-00-0

ganstigmine

509

2934 99 90

0-00-0

pitrakinra

575

2934 99 90

110299-05-3

selodenoson

365

2934 99 90

111358-88-4

lestaurtinib

686

2934 99 90

112984-60-8

ulifloxacin

676

2934 99 90

114899-77-3

trabectedin

351

2934 99 90

117276-75-2

lanimostim

776

2934 99 90

120313-91-9

thrombomodulin alfa

408

2934 99 90

120685-11-2

midostaurin

337

2934 99 90

122970-40-5

isatoribine

129

2934 99 90

123318-82-1

clofarabine

437

2934 99 90

124584-08-3

nesiritide

647

2934 99 90

130306-02-4

tezacitabine

390

2934 99 90

135306-39-7

manifaxine

130

2934 99 90

135463-81-9

coluracetam

505

2934 99 90

137071-32-0

pimecrolimus

446

2934 99 90

137215-12-4

odiparcil

812

2934 99 90

137219-37-5

plitidepsin

207

2934 99 90

143491-57-0

emtricitabine

95

2934 99 90

144348-08-3

binodenoson

474

2934 99 90

144598-75-4

paliperidone

451

2934 99 90

144689-63-4

olmesartan medoxomil (olmesartan)

33

2934 99 90

145514-04-1

amdoxovir

684

2934 99 90

145918-75-8

troxacitabine

31

2934 99 90

146426-40-6

alvocidib

585

2934 99 90

147817-50-3

siramesine

569

2934 99 90

148430-28-8

sarakalim

517

2934 99 90

150322-43-3

prasugrel

49

2934 99 90

151879-73-1

aprinocarsen

688

2934 99 90

152735-23-4

upidosin

502

2934 99 90

152811-62-6

piboserod

524

2934 99 90

153062-94-3

pumosetrag

206

2934 99 90

155030-63-0

emodepside

245

2934 99 90

159351-69-6

everolimus

382

2934 99 90

161178-07-0

lubazodone

256

2934 99 90

161605-73-8

fanapanel

609

2934 99 90

161832-65-1

talampanel

775

2934 99 90

162635-04-3

temsirolimus

704

2934 99 90

163521-12-8

vilazodone

3

2934 99 90

167362-48-3

abetimus

330

2934 99 90

169148-63-4

insulin detemir

562

2934 99 90

169939-94-0

ruboxistaurin

48

2934 99 90

170729-80-3

aprepitant

538

2934 99 90

170861-63-9

reglitazar

513

2934 99 90

171228-49-2

posaconazole

604

2934 99 90

171596-29-5

tadalafil

11

2934 99 90

171752-56-0

adrogolide

190

2934 99 90

174402-32-5

edotecarin

796

2934 99 90

174638-15-4

fosfluridine tidoxil

393

2934 99 90

176161-24-3

maribavir

417

2934 99 90

179602-65-4

mitratapid

201

2934 99 90

181785-84-2

elvucitabine

57

2934 99 90

182133-25-1

arzoxifene

5

2934 99 90

182167-02-8

acolbifene

762

2934 99 90

182415-09-4

piclozotan

289

2934 99 90

183547-57-1

gantofiban

1

2934 99 90

183849-43-6

abaperidone

293

2934 99 90

184475-35-2

gefitinib

24

2934 99 90

185229-68-9

alicaforsen

663

2934 99 90

185954-27-2

tofimilast

384

2934 99 90

187164-19-8

luliconazole

368

2934 99 90

188630-14-0

liatermin

473

2934 99 90

189681-70-7

aplindore (palindore)

148

2934 99 90

189940-24-7

daxalipram

443

2934 99 90

190977-41-4

oblimersen

309

2934 99 90

192314-93-5

iclaprim

525

2934 99 90

192374-14-4

radafaxine

379

2934 99 90

192441-08-0

lomeguatrib

516

2934 99 90

192755-52-5

pralnacasan

364

2934 99 90

193700-51-5

leridistim

68

2934 99 90

195733-43-8

atrasentan

132

2934 99 90

195962-23-3

corifollitropin alfa

258

2934 99 90

196808-45-4

farglitazar

402

2934 99 90

198821-22-6

merimepodib

456

2934 99 90

199685-57-9

onercept

191

2934 99 90

204318-14-9

edotreotide

625

2934 99 90

204512-90-3

tecadenoson

671

2934 99 90

204658-47-9

torapsel

634

2934 99 90

205887-54-3

telbermin

458

2934 99 90

206254-79-7

opebacan

334

2934 99 90

206260-33-5

irampanel

280

2934 99 90

208848-19-5

freselestat

263

2934 99 90

208993-54-8

fiduxosin

265

2934 99 90

209342-40-5

finafloxacin

154

2934 99 90

211448-85-0

denufosol

745

2934 99 90

211735-76-1

farampator

388

2934 99 90

214548-46-6

lusaperidone

814

2934 99 90

215174-50-8

rimacalib

535

2934 99 90

218298-21-6

razaxaban

543

2934 99 90

219846-31-8

radequinil (resequinil)

257

2934 99 90

221241-63-0

fandosentan

527

2934 99 90

222834-30-2

ragaglitazar

563

2934 99 90

223537-30-2

rupintrivir

99

2934 99 90

223661-25-4

bulaquine

353

2934 99 90

231277-92-2

lapatinib

359

2934 99 90

247207-64-3

leconotide

322

2934 99 90

250601-04-8

imiglitazar

8

2934 99 90

250710-65-7

adargileukin alfa

228

2934 99 90

251303-04-5

ertiprotafib

514

2934 99 90

252260-02-9

posizolid

722

2934 99 90

255730-18-8

artemifone

338

2934 99 90

257277-05-7

iseganan

104

2934 99 90

267243-28-7

canertinib

336

2934 99 90

276690-58-5

iroxanadine

651

2934 99 90

279215-43-9

tifenazoxide

118

2934 99 90

282526-98-1

cetilistat

77

2934 99 90

285571-64-4

barusiban

175

2934 99 90

285983-48-4

doramapimod

81

2934 99 90

290296-68-3

befetupitant

792

2934 99 90

292634-27-6

dianicline

615

2934 99 90

304853-42-7

tanaproget

50

2934 99 90

305391-49-5

ardenermin

771

2934 99 90

308240-58-6

talactoferrin alfa

598

2934 99 90

308831-61-0

sufugolix

537

2934 99 90

313348-27-5

regadenoson

326

2934 99 90

325715-02-4

indiplon

187

2934 99 90

328538-04-1

edifoligide

741

2934 99 90

329744-44-7

embeconazole

425

2934 99 90

331741-94-7

muraglitazar

759

2934 99 90

331744-64-0

peliglitazar

825

2934 99 90

333754-36-2

tesetaxel

635

2934 99 90

3424-98-4

telbivudine

90

2934 99 90

350992-10-8

bifeprunox

571

2934 99 90

351862-32-3

sarizotan

202

2934 99 90

361343-19-3

elzasonan

424

2934 99 90

366017-09-6

mubritinib

552

2934 99 90

366789-02-8

rivaroxaban

694

2934 99 90

380886-95-3

valtorcitabine

673

2934 99 90

40093-94-5

torcitabine

662

2934 99 90

41941-56-4

tocladesine

799

2934 99 90

434283-16-6

lecozotan

493

2934 99 90

446022-33-9

pelitrexol

339

2934 99 90

457913-93-8

ismomultin alfa

793

2934 99 90

460738-38-9

ecallantide

155

2934 99 90

506433-25-6

depelestat

414

2934 99 90

507453-82-9

mirococept

84

2934 99 90

566906-50-1

beminafil

764

2934 99 90

575458-75-2

radotermin

783

2934 99 90

583057-48-1

arasertaconazole

169

2934 99 90

59985-21-6

diquafosol

813

2934 99 90

625095-60-5

pradefovir

829

2934 99 90

640281-90-9

valopicitabine

60

2934 99 90

65576-45-6

asenapine

431

2934 99 90

84472-85-5

navuridine

559

2934 99 90

99755-59-6

rotigotine

599

2935 00 90

0-00-0

sulamserod

317

2935 00 90

123663-49-0

iguratimod

542

2935 00 90

144980-29-0

repinotan

539

2935 00 90

150375-75-0

relcovaptan

127

2935 00 90

158751-64-5

clamikalant

39

2935 00 90

161814-49-9

amprenavir

824

2935 00 90

165538-40-9

terutroban

327

2935 00 90

165668-41-7

indisulam

157

2935 00 90

169590-41-4

deracoxib

115

2935 00 90

169590-42-5

celecoxib

593

2935 00 90

170858-33-0

sonepiprazole

658

2935 00 90

174484-41-4

tipranavir

654

2935 00 90

180200-68-4

tilmacoxib

128

2935 00 90

180384-56-9

clazosentan

648

2935 00 90

180384-57-0

tezosentan

679

2935 00 90

180918-68-7

trecetilide

690

2935 00 90

181695-72-7

valdecoxib

587

2935 00 90

184036-34-8

sitaxentan

817

2935 00 90

185913-78-4

satavaptan

520

2935 00 90

192329-42-3

prinomastat

78

2935 00 90

195533-53-0

batabulin

479

2935 00 90

198470-84-7

parecoxib

145

2935 00 90

206361-99-1

darunavir

40

2935 00 90

209733-45-9

anatibant

621

2935 00 90

210538-44-6

taprizosin

189

2935 00 90

210891-04-6

edonentan

138

2935 00 90

219311-44-1

dabuzalgron

698

2935 00 90

224785-90-4

vardenafil

275

2935 00 90

226700-79-4

fosamprenavir

666

2935 00 90

233254-24-5

tomeglovir

63

2935 00 90

254877-67-3

ataciguat

123

2935 00 90

265114-23-6

cimicoxib

540

2935 00 90

266359-83-5

reparixin

827

2935 00 90

268203-93-6

udenafil

782

2935 00 90

287405-51-0

apratastat

558

2935 00 90

287714-41-4

rosuvastatin

784

2935 00 90

290815-26-8

avosentan

376

2935 00 90

321915-31-5

litomeglovir

182

2935 00 90

381683-92-7

ecopladib

739

2935 00 90

381683-94-9

efipladib

433

2935 00 90

403604-85-3

nebentan

27

2936 21 00

5300-03-8

alitretinoin

178

2936 29 90

54573-75-0

doxercalciferol

810

2937 19 00

147859-97-0

peforelin

346

2937 19 00

159768-75-9

labradimil

4

2937 19 00

178535-93-8

abrineurin

404

2937 19 00

186018-45-1

metreleptin

374

2937 19 00

204656-20-2

liraglutide

331

2937 19 00

207748-29-6

insulin glulisine

151

2937 19 00

214766-78-6

degarelix

491

2937 19 00

218620-50-9

pegvisomant

630

2937 19 00

287714-30-1

teduglutide

478

2937 19 00

345663-45-8

parathyroid hormone

719

2937 22 00

0-00-0

zoticasone

239

2937 22 00

199331-40-3

etiprednol dicloacetate

674

2937 23 00

110072-15-6

tosagestin

573

2937 23 00

7690-08-6

segesterone

687

2937 29 00

159811-51-5

uliprisnil

61

2937 29 00

199396-76-4

asoprisnil

62

2937 29 00

222732-94-7

asoprisnil ecamate

441

2937 29 00

53016-31-2

norelgestromin

43

2937 29 00

7753-60-8

anecortave

183

2937 50 00

136892-64-3

ecraprost

92

2937 50 00

155206-00-1

bimatoprost

608

2937 50 00

209860-87-7

tafluprost

816

2937 50 00

256382-08-8

rivenprost

383

2937 50 00

333963-40-9

lubiprostone

197

2937 50 00

63266-93-3

eganoprost

680

2937 50 00

81846-19-7

treprostinil

427

2939 19 00

152657-84-6

nalfurafine

756

2939 19 00

20290-10-2

morphine glucuronide

407

2939 59 00

151159-23-8

midaxifylline

340

2939 59 00

155270-99-8

istradefylline

432

2939 59 00

166374-49-8

naxifylline

247

2939 99 00

0-00-0

exatecan alideximer

246

2939 99 00

171335-80-1

exatecan

484

2939 99 00

203066-49-3

pegamotecan

12

2939 99 00

215604-75-4

afeletecan

168

2939 99 00

220997-97-7

diflomotecan

740

2939 99 00

220998-10-7

elomotecan

83

2939 99 00

256411-32-2

belotecan

298

2939 99 00

292618-32-7

gimatecan

561

2939 99 00

91421-42-0

rubitecan

607

2940 00 00

179067-42-6

tafluposide

93

2940 00 00

187269-40-5

bimosiamose

277

2940 00 00

488-69-7

fosfructose

653

2941 30 00

220620-09-7

tigecycline

313

2941 50 00

110480-13-2

idremcinal

468

2941 90 00

0-00-0

ozogamicin

244

2941 90 00

109545-84-8

evernimicin

726

2941 90 00

119673-08-4

becatecarin

113

2941 90 00

140128-74-1

cefmatilen

285

2941 90 00

140637-86-1

galarubicin

177

2941 90 00

148016-81-3

doripenem

482

2941 90 00

152044-54-7

patupilone

227

2941 90 00

153832-46-3

ertapenem

624

2941 90 00

161715-24-8

tebipenem pivoxil (tebipenem)

112

2941 90 00

162808-62-0

caspofungin

44

2941 90 00

166663-25-8

anidulafungin

348

2941 90 00

171047-47-5

ladirubicin

460

2941 90 00

171099-57-3

oritavancin

141

2941 90 00

171500-79-1

dalbavancin

636

2941 90 00

173838-31-8

telithromycin

602

2941 90 00

193811-33-5

tacapenem

117

2941 90 00

205110-48-1

cethromycin

732

2941 90 00

209467-52-7

ceftobiprole

708

2941 90 00

21102-49-8

volpristin

565

2941 90 00

211100-13-9

sabarubicin

685

2941 90 00

217500-96-4 tulathromycin A + 280755-12-6 tulath. B

tulathromycin

343

2941 90 00

219989-84-1

ixabepilone

546

2941 90 00

224452-66-8

retapamulin

114

2941 90 00

234096-34-5

cefovecin

405

2941 90 00

235114-32-6

micafungin

358

2941 90 00

371918-51-3 (component A3), 371918-44-4 (component A4)

latidectin

633

2941 90 00

372151-71-8

telavancin

733

2941 90 00

376653-43-9

ceftobiprole medocaril

693

2941 90 00

56124-62-0

valrubicin

41

3002 10 91

0-00-0

anatumomab mafenatox

217

3002 10 91

0-00-0

epitumomab

301

3002 10 91

0-00-0

hemoglobin glutamer

715

3002 10 91

0-00-0

ziralimumab

475

3002 10 91

188039-54-5

palivizumab

430

3002 10 91

189261-10-7

natalizumab

675

3002 10 91

192391-48-3

tositumomab

702

3002 10 91

195158-85-1

vepalimomab

412

3002 10 91

195189-17-4

minretumomab

400

3002 10 91

196078-29-2

mepolizumab

560

3002 10 91

197099-66-4

rovelizumab

302

3002 10 91

197462-97-8

hemoglobin raffimer

420

3002 10 91

202833-07-6

morolimumab

67

3002 10 91

202833-08-7

atorolimumab

119

3002 10 91

205923-56-4

cetuximab

221

3002 10 91

205923-57-5

epratuzumab

306

3002 10 91

206181-63-7

ibritumomab tiuxetan

225

3002 10 91

211323-03-4

erlizumab

459

3002 10 91

213327-37-8

oregovomab

96

3002 10 91

214559-60-1

bivatuzumab

194

3002 10 91

214745-43-4

efalizumab

20

3002 10 91

216503-57-0

alemtuzumab

418

3002 10 91

216503-58-1

mitumomab

581

3002 10 91

216669-97-5

sibrotuzumab

86

3002 10 91

216974-75-3

bevacizumab

345

3002 10 91

219649-07-7

labetuzumab

185

3002 10 91

219685-50-4

eculizumab

501

3002 10 91

219685-93-5

pexelizumab

706

3002 10 91

219716-33-3

visilizumab

297

3002 10 91

220578-59-6

gemtuzumab

564

3002 10 91

220651-94-5

ruplizumab

620

3002 10 91

235428-87-2

taplitumomab paptox

545

3002 10 91

241473-69-8

reslizumab

453

3002 10 91

242138-07-4

omalizumab

292

3002 10 91

244096-20-6

gavilimomab

360

3002 10 91

250242-54-7

lemalesomab

670

3002 10 91

252662-47-8

toralizumab

218

3002 10 91

263547-71-3

epitumomab cituxetan

47

3002 10 91

267227-08-7

apolizumab

403

3002 10 91

272780-74-2

metelimumab

363

3002 10 91

285985-06-0

lerdelimumab

584

3002 10 91

288392-69-8

siplizumab

184

3002 10 91

292819-64-8

ecromeximab

639

3002 10 91

299423-37-3

teneliximab

274

3002 10 91

326859-36-3

fontolizumab

480

3002 10 91

331243-22-2

pascolizumab

7

3002 10 91

331731-18-1

adalimumab

697

3002 10 91

336801-86-6

vapaliximab

477

3002 10 91

339177-26-3

panitumumab

395

3002 10 91

339186-68-4

matuzumab

530

3002 10 91

347396-82-1

ranibizumab

82

3002 10 91

356547-88-1

belimumab

286

3002 10 91

357613-77-5

galiximab

385

3002 10 91

357613-86-6

lumiliximab

85

3002 10 91

375348-49-5

bertilimumab

661

3002 10 91

375823-41-9

tocilizumab

612

3002 10 91

380610-22-0

talizumab

499

3002 10 91

380610-27-5

pertuzumab

59

3002 10 91

395639-53-9

aselizumab

106

3002 10 91

400010-39-1

cantuzumab mertansine

116

3002 10 91

428863-50-7

certolizumab pegol

200

3002 10 91

468715-71-1

elsilimomab

300

3002 10 91

476181-74-5

golimumab

521

3002 10 91

499212-74-7

pritumumab

689

3002 10 91

502496-16-4

urtoxazumab

9

3002 10 91

503605-66-1

adecatumumab

789

3002 10 91

509077-98-9

catumaxomab

794

3002 10 91

509077-99-0

ertumaxomab

774

3002 10 91

521079-87-8

tefibazumab

729

3002 10 91

537694-98-7

besilesomab

830

3002 10 91

558480-40-3

volociximab

765

3002 10 91

565451-13-0

raxibacumab

369

3002 10 91

569658-79-3

libivirumab

248

3002 10 91

569658-80-6

exbivirumab

808

3002 10 91

595566-61-3

pagibaximab

751

3002 10 91

635715-01-4

inotuzumab ozogamicin

785

3002 10 91

648895-38-9

bapineuzumab

713

3002 10 91

652153-01-0

zanolimumab

802

3002 10 91

658052-09-6

mapatumumab

832

3002 10 91

667901-13-5

zalutumumab

805

3002 10 91

679818-59-8

ofatumumab

319

3002 10 95

149824-15-7

ilodecakin

42

3002 10 95

163545-26-4

ancestim

236

3002 10 95

185243-69-0

etanercept

188

3002 10 95

187348-17-0

edodekin alfa

94

3002 10 95

207137-56-2

binetrakin

143

3002 10 95

209810-58-2

darbepoetin alfa

18

3002 10 95

222535-22-0

alefacept

415

3002 10 95

244130-01-6

mirostipen

291

3002 10 95

246861-96-1

garnocestim

220

3002 10 95

261356-80-3

epoetin delta

2

3002 10 95

332348-12-6

abatacept

617

3002 10 95

465540-87-8

taneptacogin alfa

749

3002 10 95

479198-61-3

iboctadekin

742

3002 10 95

604802-70-2

epoetin zeta

786

3002 10 95

706808-37-9

belatacept

179

3002 10 95

98530-76-8

drotrecogin alfa (activated)

780

3002 10 99

84720-88-7

antithrombin alfa

70

3002 90 90

223577-45-5

aviscumine

734

3002 90 90

372075-36-0

cintredekin besudotox

779

3504 00 00

9009-65-8

protamine sulfate

243

3507 90 90

0-00-0

eufauserase

13

3507 90 90

104138-64-9

agalsidase alfa

14

3507 90 90

104138-64-9

agalsidase beta

533

3507 90 90

134774-45-1

rasburicase

429

3507 90 90

136653-69-5

nasaruplase beta

160

3507 90 90

145137-38-8

desmoteplase

34

3507 90 90

151912-11-7

amediplase

638

3507 90 90

191588-94-0

tenecteplase

532

3507 90 90

196488-72-9

ranpirnase

216

3507 90 90

208576-22-1

epafipase

356

3507 90 90

210589-09-6

laronidase

22

3507 90 90

259074-76-5

alfimeprase

23

3507 90 90

420784-05-0

alglucosidase alfa

315

3507 90 90

50936-59-9

idursulfase (idusulfase)

747

3507 90 90

552858-79-4

galsulfase

748

3507 90 90

9074-87-7

glucarpidase

426

3906 90 90

246527-99-1

mureletecan

485

3907 20 21

0-00-0

pegaptanib

483

3907 20 21

187139-68-0

pegacaristim

487

3907 20 21

198153-51-4

peginterferon alfa-2a

489

3907 20 21

204565-76-4

pegnartograstim

486

3907 20 21

208265-92-3

pegfilgrastim

488

3907 20 21

215647-85-1

peginterferon alfa-2b

490

3907 20 21

330988-75-5

pegsunercept

470

3908 90 00

263351-82-2

paclitaxel poliglumex

664

3911 90 99

28210-41-5

tolevamer

377

3913 90 00

329306-27-6

livaraparin calcium

152

3913 90 00

9041-08-1

deligoparin sodium

(1)  Commission Regulation (EC) No 1549/2006 of 17 October 2006 amending Annex I to Council Regulation (EEC) No 2658/87 on the tariff and statistical nomenclature and on the Common Customs Tariff (
OJ L 301, 31.10.2006, p. 1
).

ANNEX II

List of prefixes and suffixes which, in combination with the INNs of Annex 3 to Regulation (EC) No 1549/2006, describe the salts, esters or hydrates of INNs; these salts, esters and hydrates are free of duty, on condition that they are classifiable in the same six-digit HS-subheading as the corresponding INN

Prefixes and suffixes can be combined (e.g. hydrochloride phosphate). They can be preceded by a multiplying prefix such as bi, bis, di, hemi, hepta, hexa, mono, penta, sesqui, tetra, tri, tris… (e.g. diacetate). Synonyms and systematic names can also be used, in the same way.
INN means International Nonproprietary Names for pharmaceutical substances, World Health Organisation.
INNRG means International Nonproprietary Names (INN) for pharmaceutical substances, Names for radicals & groups, comprehensive list 2004.
INNCN means chemical or systematic name listed in International Nonproprietary Names (INN) for pharmaceutical substances, Names for radicals & groups, comprehensive list 2004.

ID

Preferred prefix or suffix

Synonyms

Systematic name when different

1

acefurate (INNRG)

 

acetate (ester), furan-2-carboxylate (ester) (INNCN)

2

aceglumate (INNRG)

 

rac-hydrogen N-acetylglutamate (INNCN)

3

aceponate (INNRG)

 

acetate (ester), propanoate (ester) (INNCN)

4

acetate

 

 

5

acetonide (INNRG)

 

propane-2,2-diylbis(oxy) (INNCN)

6

acetofenide

acetophenide

1-phenylethane-1,1-diylbis(oxy)

7

1-acetoxyethyl

 

1-(acetyloxy)ethyl

8

aceturate (INNRG)

 

N-acetylglycinate (INNCN)

10

acetylsalicylate

 

2-(acetyloxy)benzoate

11

acibutate (INNRG)

 

acetate (ester), 2-methylpropanoate (ester) (INNCN)

12

acistrate (INNRG)

 

acetate (ester), octadecanoate (ester) (INNCN)

13

acoxil (INNRG)

 

(acetyloxy)methyl (INNCN)

14

adipate

 

hexanedioate

15

alfoscerate (INNRG)

 

(2R)-2,3-dihydroxypropyl hydrogen phosphate (INNCN)

16

alideximer (INNRG)

 

poly([oxy(2-hydroxyethane-1,1-diyl)]{oxy[1-(hydroxymethyl)ethane-1,2-diyl]}) partly O-etherified with carboxymethyl groups with some carboxy groups amide linked to the tetrapeptide residue (glycylglycyl-L-phenylalanylglycyl) (INNCN)

17

allyl

 

prop-2-en-1-yl

18

allylbromide

allylobromide

N-allyl, bromide (salt)

19

allyliodide

allyloiodide

N-allyl, iodide (salt)

20

aluminium

 

 

21

4-aminosalicylate

aminosalicylate

2-hydroxy-4-aminobenzoate

22

ammonium

 

 

24

amsonate (INNRG)

 

2,2'-ethene-1,2-diylbis (5-aminobenzene-1-sulfonate) (INNCN)

25

anisatil (INNRG)

 

2-(4-methoxyphenyl)-2-oxoethyl (INNCN)

26

antipyrate

 

 

27

arbamel (INNRG)

 

2-(dimethylamino)-2-oxoethyl (INNCN)

28

argine (INNRG)

 

30Bα-L-arginine-30Bβ-L-arginine (INNCN)

29

arginine (INN)

 

 

30

aritox (INNRG)

 

ricin A chain-MAB immunotoxine (INNCN)

31

ascorbate

 

 

32

aspart (INNRG)

 

28B-L-aspartic acid- (INNCN)

33

aspartate

 

 

34

axetil (INNRG)

 

rac-1-(acetyloxy)ethyl (INNCN)

35

barbiturate

 

2,4,6(1H,3H,5H)-pyrimidinetrione

36

benetonide (INNRG)

 

N-benzoyl-2-methyl-β-alanine (ester), acetonide (INNCN)

37

benzathine

 

N,N'-dibenzylethylenediammonium

40

benzoacetate

 

 

41

benzoate (INNRG)

 

 

42

benzyl

 

 

43

benzylbromide

benzylobromide

N-benzyl, bromide (salt)

44

benzyliodide

benzyloiodide

N-benzyl, iodide (salt)

45

besilate (INNRG)

besylate

benzenesulfonate (INNCN), benzenesulphonate

47

bezomil (INNRG)

 

(benzoyloxy)methyl (INNCN)

53

bismuth

 

 

55

borate

 

 

56

bromide (INNRG)

 

 

57

buciclate (INNRG)

 

trans-4-butylcyclohexanecarboxylate (INNCN)

58

bunapsilate (INNRG)

 

3,7-di-tert-butylnaphthalene-1,5-disulfonate (INNCN)

59

buteprate (INNRG)

 

butyrate (ester), propionate (ester) (INNCN)

60

butyl

 

 

62

tert-butyl

t-butyl, tertiary butyl

 

67

butyl ester

 

 

69

tert-butyl ester

t-butyl ester, tertiary butyl ester

 

75

butylbromide

butylobromide

N-butyl, bromide (salt)

76

butyrate

butylate

butanoate

77

calcium

 

 

82

camphorate

 

1,2,2-trimethyl-1,3-cyclopentanedicarboxylate

85

camsilate (INNRG)

camsylate, camphorsulfonate, camphorsulphonate, R-camphorsulfonate, R-camphorsulphonate, S-camphorsulfonate, S-camphorsulphonate, camphor-10-sulfonate, camphor-10-sulphonate

(7,7-dimethyl-2-oxobicyclo[2.2.1]heptan-1-yl)methanesulfonate (INNCN)

87

caproate (INNRG)

 

hexanoate (INNCN)

88

carbamate

 

 

89

carbesilate (INNRG)

 

4-sulfobenzoate (INNCN)

90

carbonate

 

 

91

chloride (INNRG)

 

 

95

choline

 

(2-hydroxyethyl)trimethylammonium

96

ciclotate (INNRG)

cyclotate

4-methylbicyclo[2.2.2]oct-2-ene-1-carboxylate (INNCN)

97

cilexetil (INNRG)

 

rac-1-{[(cyclohexyloxy)carbonyl]oxy}ethyl (INNCN)

98

cinnamate

 

3-phenylprop-2-enoate

99

cipionate (INNRG)

cypionate, cyclopentanepropionate

3-cyclopentylpropanoate (INNCN), 3-cyclopentylpropionate

100

citrate

 

2-hydroxypropane-1,2,3-tricarboxylate

101

cituxetan (INNRG)

 

N-(4-{2(RS)-2-[bis(carboxymethyl)amino)]-3-({2-[bis(carboxymethyl)=amino]ethyl}(carboxymethyl)amino)propyl}phenyl)thiocarbamoyl (INNCN)

102

clofibrol (INNRG)

 

2-(4-chlorophenoxy)-2-methylpropyl (INNCN)

103

closilate (INNRG)

closylate, p-chlorobenzenesulfonate, p-chlorobenzenesulphonate

4-chlorobenzene-1-sulfonate (INNCN), 4-chlorobenzenesulfonate

105

crobefate (INNRG)

 

rac-{3-[(3E)-4-methoxybenzylidene]-2-(4-methoxyphenyl)chroman- 6-yl phosphate(2-)} (INNCN)

106

cromacate (INNRG)

 

2-[(6-hydroxy-4-methyl-2-oxo-2H-chromen-7yl)oxy]acetate (INNCN)

107

cromesilate (INNRG)

 

(6,7-dihydroxy-2-oxo-2H-chromen-4-yl)methanesulfonate (INNCN)

108

crosfumaril (INNRG)

 

(2E)-but-2-enedioyl (INNCN)

109

cyclamate (INNRG)

N-cyclohexylsulfamate, N-cyclohexylsulphamate

cyclohexylsulfamate (INNCN)

110a

cyclohexylamine

 

 

111

cyclohexylammonium

 

 

112

cyclohexylpropionate

cyclohexanepropionate

cyclohexylpropanoate

118

daloxate (INNRG)

 

L-alaninate (ester), (5-methyl-2-oxo-1,3-dioxol-4-yl)methyl (INNCN)

120

daropate (INNRG)

dapropate

3-(dimethylamino)propanoate (INNCN)

121

deanil (INNRG)

 

2-(dimethylamino)ethyl (INNCN)

122

decanoate

 

 

123

decil (INNRG)

 

decyl (INNCN)

124

defalan (INNRG)

 

des-1B-L-phenylalanine-insulin (INNCN)

125

detemir (INNRG)

 

tetradecanoyl (INNCN)

129

dibudinate (INNRG)

 

2,6-di-tert-butylnaphthalene-1,5-disulfonate (INNCN)

130

dibunate (INNRG)

 

2,6-di-tert-butylnaphthalene-1-sulfonate (INNCN)

133

dicibate (INNRG)

 

dicyclohexylmethyl carbonate (INNCN)

134

dicyclohexylamine

 

 

135

dicyclohexylammonium

 

 

137

diethylamine

 

 

138

diethylammonium

 

 

139

diftitox (INNRG)

 

N-L-methionyl-387-L-histidine-388-L-alanine-1-388-toxin (Corynebacterium diphtheriae strain C7) (388→2')-protein (INNCN)

142

digolil (INNRG)

 

2-(2-hydroxyethoxy)ethyl (INNCN)

149

dihydroxybenzoate

 

 

154

N,N-dimethyl-β-alanine

N,N-dimethyl-beta-alanine

 

156

dinitrobenzoate

 

 

157

diolamine (INNRG)

diethanolamine

2,2'-azanediyldiethanol (INNCN)

165

disulfide

disulphide

 

169

docosil (INNRG)

 

docosyl (INNCN)

170

dofosfate (INNRG)

 

octadecyl hydrogen phosphate (INNCN)

171

ecamate (INNRG)

 

N-ethylcarbamate (INNCN)

172

edamine (INNRG)

 

ethane-1,2-diamine (INNCN)

173

edisilate (INNRG)

edisylate, 1,2-ethanedisulfonate, 1,2-ethanedisulphonate

ethane-1,2-disulfonate (INNCN)

175

embonate (INNRG)

pamoate, 4,4'-methylenebis(3-hydroxy-2-naphthoate)

4,4'-methylenebis(3-hydroxynaphthalene-2-carboxylate) (INNCN)

176

enantate (INNRG)

enanthate

heptanoate (INNCN)

178

enbutate (INNRG)

 

acetate (ester), butanoate (ester) (INNCN)

179

epolamine (INNRG)

1-pyrrolidineethanol

2-(pyrrolidin-1-yl)ethanol (INNCN)

180

erbumine (INNRG)

tert-butylamine, t-butylamine, tertiary butylamine

2-methylpropan-2-amine (INNCN)

181

esilate (INNRG)

esylate, ethanesulfonate, ethanesulphonate

ethanesulfonate (INNCN)

182

estolate (INNRG)

propionate dodecyl sulfate, propionate dodecyl sulphate, propionate lauryl sulfate, propionate lauryl sulphate

propanoate (ester), dodecyl sulfate (salt) (INNCN)

184

etabonate (INNRG)

 

ethyl carbonate (INNCN)

190

ethylbromide

ethobromide

N-ethyl, bromide (salt)

191

ethyl

 

 

192

ethyl ester

 

 

193

ethylamine

 

 

194

ethylammonium

 

 

195

ethylenantate

ethylheptanoate

 

196

ethylenediamine

 

ethane-1,2-diamine

197

ethylhexanoate

 

 

198

ethyliodide

ethyloiodide

N-ethyl, iodide (salt)

199

ethylsuccinate

 

 

200

etilsulfate (INNRG)

ethylsulfate

ethyl sulfate (INNCN)

201

farnesil (INNRG)

 

(2E,6E)-3,7,11-trimethyldodeca-2,6,10-trien-1-yl (INNCN)

202

fendizoate (INNRG)

 

2-(6-hydroxybiphenyl-3-carbonyl)benzoate (INNCN)

203a

ferrous

 

 

204

fluoride

 

 

205

fluorosulfonate

fluorosulphonate

 

207

formate

 

 

209

fosfatex

 

 

210

fostedate (INNRG)

 

tetradecyl hydrogen phosphate (INNCN)

211

fumarate

 

(2E)-but-2-enedioate

212

furetonide (INNRG)

 

1-benzofurane-2-carboxylate (ester), propane-2,2-diylbis(oxy) (INNCN)

213

furoate

 

furan-2(or 3)-carboxylate

213a

fusidate

 

 

214

gadolinium

 

 

215

gamolenate (INNRG)

 

(6Z,9Z,12Z)-octadeca-6,9,12-trienoate (INNCN)

216

glargine (INNRG)

 

21A-glycine-30Bα-L-arginine-30Bβ-L-arginine (INNCN)

217

glucarate

saccharate

(2R,3S,4S,5S)-2,3,4,5-tetrahydroxyhexanedioate, D-glucarate

218

gluceptate (INNRG)

glucoheptonate

D-glycero-D-gulo-heptonate (INNCN)

220

gluconate

 

 

221

glucoside

 

 

222

glulisine (INNRG)

 

3B-L-lysine,29B-L-glutamic acid (INNCN)

223

glutamer (INNRG)

 

glutaraldehyde polymer (INNCN)

224

glycolate

 

hydroxyacetate

225

glyoxylate

 

oxoacetate

226

gold

 

 

227

guacil (INNRG)

 

2-methoxyphenyl (INNCN)

228

guanidine

 

 

230

hemisuccinate (INNRG)

hydrogen succinate

hydrogen butanedioate (INNCN)

235

hexacetonide (INNRG)

 

3,3-dimethylbutanoate (ester), propan-2,2-diylbis(oxy) (INNCN)

238

hibenzate (INNRG)

hybenzate

4-(4-hydroxybenzoyl)benzoate (INNCN)

239

hippurate

 

N-Benzoylglycine salt

241

hyclate (INNRG)

 

ethanol — hydrogen chloride — water (0,5 /1/0,5 ) (INNCN)

242

hydrate

 

 

243

hydrobromide

 

 

244

hydrochloride

 

 

248a

hydrogen

 

 

261

hydroxide

 

 

262

hydroxybenzoate

 

 

263

2-(4-hydroxybenzoyl)benzoate

o-(4-hydroxybenzoyl)benzoate

 

267

hydroxynaphtoate (INNRG)

hydroxynaphthoate

3-hydroxynaphthalene-2-carboxylate (INNCN)

268

iodide (INNRG)

 

 

269

iodine-131

 

 

270

iron chloride

 

 

272

isetionate (INNRG)

isethionate, 2-hydroxyethansulfonate, 2-hydroxyethansulphonate

2-hydroxyethane-1-sulfonate (INNCN)

273

isobutyrate

 

2-methylpropanoate

274

isocaproate

 

4-methylpentanoate

275

isonicotinate

 

pyridine-4-carboxylate

276

isophthalate

 

benzene-1,3-dicarboxylate

277

isopropionate

 

 

278

isopropyl

 

propan-2-yl

279

lactate

 

2-hydroxypropanoate

280

lactobionate

 

4-O-(β-D-galactopyranosyl)-D-gluconate

281

laurate (INNRG)

 

dodecanoate (INNCN)

282

lauril (INNRG)

lauryl

dodecyl (INNCN)

283

laurilsulfate (INNRG)

lauril sulfate, lauril sulphate, lauryl sulfate, lauryl sulphate, laurilsulphate, laurylsulfate, laurylsulphate

dodecyl sulfate (INNCN)

288

levulinate

 

4-oxopentanoate

289

lisetil (INNRG)

 

L-lysinate (ester), diethyl (ester) (INNCN)

290

lisicol (INNRG)

 

{N-[(5S)-5-carboxy-5-(3α,7α,12α-trihydroxy-5β-cholan-24-amido)pentyl]carbamothioyl}amino (INNCN)

291

lispro (INNRG)

 

28B-L-lysine-29B-L-proline (INNCN)

292

lithium

 

 

293

lutetium

 

 

294

lysinate

lysine (INN)

 

296

mafenatox (INNRG)

 

enterotoxin A (227-alanine) (Staphylococcus aureus) (INNCN)

297

magnesium

 

 

298

malate

 

hydroxybutanedioate

299

maleate

 

(Z)-but-2-enoate

300

malonate

 

propanedioate

301

mandelate

 

2-hydroxy-2-phenylacetate, α-hydroxybenzeneacetate

302

medoxomil (INNRG)

 

(5-methyl-2-oxo-1,3-dioxol-4-yl)methyl (INNCN)

303

megallate (INNRG)

 

3,4,5-trimethoxybenzoate (INNCN)

304

meglumine (INN)

N-methylglucamine

1-deoxy-1-methylamino-D-glucitol

305

merpentan (INNRG)

 

{N,N'-[1-(3-oxopropyl)ethane-1,2-diyl]bis(2-sulfanylacetamidato)}(4-) (INNCN)

306

mertansine (INNRG)

 

tetrakis{(4RS)-4[(3-{[(1S)-2-{[(1S,2R,3S,5S,6S,16E,18E,20R,21S)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl]oxy}-1-methyl-2-oxoethyl]methylamino}-3-oxopropyl)disulfanyl]pentanoyl} (INNCN)

307

mesilate (INNRG)

mesylate, methanesulfonate, methanesulphonate

methanesulfonate (INNCN)

309

metembonate (INNRG)

 

4,4'-methylenebis(3-methoxynaphthalene-2-carboxylate) (INNCN)

312

methonitrate (INNRG)

 

N-methyl, nitrate (salt) (INNCN)

313

methyl ester

 

 

315

methylbromide (INNRG)

methobromide

N-methyl, bromide (salt) (INNCN)

317

methylenedisalicylate

 

methylenebis(2-hydroxybenzoate)

322

metilsulfate (INNRG)

metilsulphate, methylsulfate, methylsulphate

methyl sulfate (INNCN)

324

metiodide (INNRG)

methyliodide

N-methyl, iodide (salt) (INNCN)

325

mofetil (INNRG)

 

2-(morpholin-4-yl)ethyl (INNCN)

330

mucate

galactarate, meso-galactarate

2,3,4,5-tetrahydroxyhexane-1,6-dioate

331

nafate

formate sodium

formyloxy (ester), sodium (salt)

332

napadisilate (INNRG)

napadisylate, 1,5-naphthalenedisulfonate, 1,5-naphthalenedisulphonate

naphthalene-1,5-disulfonate (INNCN)

338

napsilate (INNRG)

napsylate, 2-naphthalenesulfonate, 2-naphthalenesulphonate

naphthalene-2-sulfonate (INNCN)

340

nicotinate (INNRG)

 

pyridine-3-carboxylate (INNCN)

341

nitrate

 

 

342

nitrobenzoate

 

 

343

octil (INNRG)

 

octyl (INNCN)

344

olamine (INNRG)

ethanolamine

2-aminoethanol (INNCN)

345

oleate (INNRG)

 

(9Z)-octadec-9-enoate (INNCN)

346

orotate

 

1,2,3,6-tetrahydro-2,6-dioxopyrimidine-4-carboxylate

348

oxalate

 

 

349

oxide

 

 

351

oxoglurate (INNRG)

 

hydrogen 2-oxopentanedioate (INNCN)

353

palmitate (INNRG)

 

hexadecanoate (INNCN)

356

pantothenate

 

N-(2,4-dihydroxy-3,3-dimethyl-1-oxobutyl)-β-alaninate

359

pegol (INNRG)

 

α-(2-carboxyethyl)-ω-methoxypoly(oxyethane-1,2-diyl) (INNCN)

360

pendetide (INN)

 

 

362

pentexil (INNRG)

pivetil

(RS)-1-[(2,2-dimethylpropanoyl)oxy]ethyl (INNCN)

363

perchlorate (INNRG)

 

 

364

phenylpropionate

 

 

365

phosphate

orthophosphate

 

366

phosphite

 

 

367

phthalate

 

benzene-1,2-dicarboxylate

368

picrate

 

2,4,6-trinitrobenzene-1-olate

369

pivalate (INNRG)

trimethylacetate

2,2-dimethylpropanoate (ester) (INNCN)

371

pivoxetil (INNRG)

 

rac-1-[(2-methoxy-2-methylpropanoyl)oxy]ethyl (INNCN)

372

pivoxil (INNRG)

(pivaloyloxy)methyl

[(2,2-dimethylpropanoyl)oxy]methyl (INNCN)

374

poliglumex (INNRG)

 

[poly(L-glutamic acid)z—(L-glutamate-γ-ester)—poly(L-glutamic acid)y]n (INNCN)

375

potassium (INNRG)

 

potassium (INNCN)

378

propionate

 

propanoate

383

propyl

 

 

384

propyl ester

 

 

385

proxetil (INNRG)

 

rac-1-{[(propan-2-yloxy)carbonyl]oxy}ethyl (INNCN)

386

pyridylacetate

 

pyridinylacetate

388

quinate

 

1,3,4,5-tetrahydroxycyclohexanecarboxylate

389

raffimer (INNRG)

 

(2S,4R,6R,8S,11S,13S)-2,4,8,13-tetrakis(hydroxymethyl)-4,6,11-tris(ylomethyl)-3,5,7,10,12-pentaoxatetradecane-1,14-diyl (INNCN)

390

resinate

abietate

(1R,4aR,4bR,10aR)-1,4a-dimethyl-7-(1-methylethyl)-1,2,3,4,4a,4b,5,6,10,10a-decahydro-1-phenanthrenecarboxylate

392

salicylate (INNRG)

 

2-hydroxybenzoate (INNCN)

393

salicyloylacetate

 

2-hydroxybenzoylacetate

394

sesquioleate (INNRG)

 

(9Z)-octadec-9-enoate(1,5) (INNCN)

395

sodium (INNRG)

 

 

413

soproxil (INNRG)

 

{[(propan-2-yloxy)carbonyl]oxy}methyl (INNCN)

414

steaglate (INNRG)

 

2-(octadecanoyloxy)acetate (ester) (INNCN)

415

stearate (INNRG)

 

octadecanoate (INNCN)

416

stinoprate (INNRG)

 

N-acetylcysteinate (salt), propanoate (ester) (INNCN)

417

succinate

 

butanedioate

418

succinil (INNRG)

 

3-carboxypropanoyl (INNCN)

419

succinyl

 

butanedioyl

420

sudotox (INNRG)

 

248-L-histidine-249-L-methionine-250-L-alanine-251-L-glutamic acid-248-613-exotoxin A (Pseudomonas aeruginosa reduced) (INNCN)

421

suleptanate (INNRG)

 

8-[methyl(2-sulfoethyl)amino]-8-oxooctanoate (ester), monosodium salt (INNCN)

422

sulfate (INNRG)

sulphate

 

423

sulfinate

sulphinate

 

424

sulfite

sulphite

 

424a

sulfobenzoate

sulphobenzoate

 

424b

3-sulfobenzoate

3-sulphobenzoate

 

425

sulfosalicylate

sulphosalicylate

2-hydroxysulfobenzoate

426

sulfoxylate (INNRG)

 

sulfinomethyl, monosodium salt (INNCN)

431

tafenatox (INNRG)

 

enterotoxin A (Staphyloccus aureus) (INNCN)

432

tannate

 

 

433

tartrate (INNRG)

L-tartrate

(2R,3R)-2,3-dihydroxybutanedioate (INNCN), L-tartarate

434

D-tartrate

 

(2S,3S)-2,3-dihydroxybutanedioate, D-tartarate

435

tebutate (INNRG)

tert-butylacetate, t-butyl acetate, tertiary butyl acetate

3,3-dimethylbutanoate (INNCN)

436

tenoate (INNRG)

 

thiophene-2-carboxylate (INNCN)

437

teoclate (INNRG)

theoclate, 8-chlorotheophyllinate

8-chloro-1,3-dimethyl-2,6-dioxo-3,6-dihydro-1H-purin-7-(2H)-ide (INNCN)

438

teprosilate (INNRG)

 

3-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-7H-purin-7-yl)propane-1-sulfonate (INNCN)

441

tetrahydrophthalate

 

cyclohexene-1,2-dicarboxylate

444

tetraxetan (INNRG)

 

[4,7,10-tris(carboxymethyl)-1,4,7,10-tetraazacyclodec-1-yl]acetyl (INNCN)

446

thiocyanate

 

 

447

tidoxil (INNRG)

 

rac-2-(decyloxy)-3-(dodecylsulfanyl)propyl (INNCN)

448

tiuxetan (INNRG)

 

N-(4-{(2S)-2-[bis(carboxymethyl)amino]-3-[(2RS)-{2-[bis(carboxymethyl)amino]propyl (carboxymethyl)amino]propyl} phenyl) thiocarbamoyl (INNCN)

449

tocoferil (INNRG)

 

rac-(2R)-2,5,7,8-tetramethyl-2-[(4R,8R)-4,8,12-trimethyltridecyl]chroman-6-yl (INNCN)

450

tofesilate (INNRG)

 

3-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-7H-purin-7-yl)ethane-1-sulfonate (INNCN)

453

tosilate (INNRG)

tosylate, p-toluenesulfonate, p-toluenesulphonate

4-methylbenzene-1-sulfonate (INNCN)

455

triclofenate (INNRG)

 

2,4,5-trichlorophenolate (INNCN)

458

triflutate (INNRG)

 

trifluoroacetate (INNCN)

463

trioleate (INNRG)

 

tris[(9Z)-octadec-9-enoate] (INNCN)

465

tristearate (INNRG)

 

tris(octadecanoate) (INNCN)

466

trolamine (INNRG)

triethanolamine

2,2',2''-nitrilotriethanol (INNCN)

467

trometamol (INN)

tromethamine

2-amino-2-(hydroxymethyl)propane-1,3-diol, tris(hydroxymethyl)methylamine

469

troxundate (INNRG)

 

[2-(2-ethoxyethoxy)ethoxy]acetate (INNCN)

472

undecylate (INNRG)

 

undecanoate (INNCN)

473

undecylenate (INNRG)

 

undec-10-enoate (INNCN)

474

valerate (INNRG)

 

pentanoate (INNCN)

475

xinafoate (INNRG)

 

1-hydroxynaphthalene-2-carboxylate (INNCN)

476

zinc

 

 

ANNEX III

List of pharmaceutical intermediates, i.e. compounds used for the manufacture of finished pharmaceutical products, to be added to the list of products receiving duty-free treatment included in Annex 6 to Regulation (EC) No 1549/2006

ID No

CN code

CAS RN

Name

793

2902 19 80

6746-94-7

ethynylcyclopropane

397

2905 29 90

173200-56-1

(E)-6,6-dimethylhept-2-en-4-yn-1-ol

250

2905 59 99

60827-45-4

(2S)-3-chloropropane-1,2-diol

320

2906 29 00

127852-28-2

(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethan-1-ol

308

2906 29 00

167155-76-2

1,1-difluoro-1,1a,6,10b-tetrahydrodibenzo[a, e]cyclopropa[c][7]annulen-6-ol

530A

2909 30 38

3259-03-8

1-(2-bromoethoxy)-2-ethoxybenzene or 2-bromoethyl 2-ethoxyphenyl ether

3

2909 30 90

165254-21-7

1,2-bis{2-[2-(2-methoxyethoxy)ethoxy]ethoxy}-4,5-dinitrobenzene

124

2909 49 90

170277-77-7

(3S)-3-[2-(mesyloxy)ethoxy]-4-(trityloxy)butyl methanesulfonate

636

2913 00 00

80565-30-6

4'-chlorobiphenyl-4-carbaldehyde

566

2914 50 00

17720-60-4

1-(2,4-dihydroxyphenyl)-2-(4-hydroxyphenyl)ethan-1-one

17

2914 50 00

4495-66-3

1-[4-(benzyloxy)phenyl]propan-1-one

316

2914 50 00

82499-20-5

(1R)-1-hydroxy-1-(3-hydroxyphenyl)acetone

712

2914 70 00

124379-29-9

(4S)-4-(3,4-dichlorophenyl)-3,4-dihydronaphthalen-1(2H)-one

43

2914 70 00

135306-45-5

1-(3,5-difluorophenyl)propan-1-one

59

2914 70 00

162548-73-4

4,6-difluoroindan-1-one

158

2914 70 00

190965-45-8

(2-bromo-5-propoxyphenyl)(2-hydroxy-4-methoxyphenyl)methanone

863

2914 70 00

2196-99-8

2-chloro-1-(4-methoxyphenyl)ethan-1-one

314

2914 70 00

2350-46-1

1-(2,3-dichloro-4-hydroxyphenyl)butan-1-one

827

2914 70 00

26771-69-7

2-methoxy-1-[4-(trifluoromethyl)phenyl]ethan-1-one

550

2914 70 00

43229-01-2

1-[4-(benzyloxy)-3-nitrophenyl]-2-bromoethan-1-one

64

2914 70 00

62932-94-9

2-bromo-1-[4-hydroxy-3-(hydroxymethyl)phenyl]ethan-1-one

755

2915 39 80

2243-35-8

2-oxo-2-phenylethyl acetate

519

2915 39 80

60176-77-4

(1S,4R)-4-hydroxycyclopent-2-en-1-yl acetate

418

2915 50 00

158894-67-8

1-bromo-2-methylpropyl propionate

796

2915 90 20

7693-41-6

4-methoxyphenyl chloroformate

686

2916 20 00

122665-97-8

4,4-difluorocyclohexane-1-carboxylic acid

937

2916 39 00

114772-40-6

tert-butyl 4'-(bromomethyl)biphenyl-2-carboxylate

869

2916 39 00

1716-12-7

sodium 4-phenylbutanoate

444

2916 39 00

2444-36-2

(2-chlorophenyl)acetic acid

394

2916 39 00

2901-13-5

ethyl 2-methyl-2-phenylpropanoate

67

2918 19 85

111969-64-3

(1R,2S,5R)-2-isopropyl-5-methylcyclohexyl dihydroxyacetate or thymol glyoxylate

760

2918 19 85

138-59-0

(3R,4S,5R)-3,4,5-trihydroxycyclohex-1-ene-1-carboxylic acid

544

2918 19 85

20585-34-6

(2S)-cyclohexyl(hydroxy)phenylacetic acid

545

2918 19 85

4335-77-7

cyclohexyl(hydroxy)phenylacetic acid

445

2918 19 85

52950-18-2

(2R)-(2-chlorophenyl)hydroxyacetic acid

508

2918 30 00

134176-18-4

ethyl 2-oxobicyclo[3.1.0]hexane-6-carboxylate

214

2918 30 00

149437-76-3

5-(4-fluorophenyl)-5-oxopentanoic acid

21

2918 30 00

39562-16-8

ethyl (E)-2-(3-nitrobenzylidene)-3-oxobutanoate

20

2918 30 00

39562-22-6

2-methoxyethyl (E)-2-(3-nitrobenzylidene)-3-oxobutanoate

23

2918 30 00

39562-27-1

methyl (2E)-2-(2-nitrobenzylidene)-3-oxobutanoate

315

2918 99 90

1217-67-0

(4-butyryl-2,3-dichlorophenoxy)acetic acid

108

2918 99 90

13335-71-2

(2,6-dimethylphenoxy)acetic acid

532

2918 99 90

150726-89-9

dimethyl (2-methoxyphenoxy)malonate

402

2918 99 90

204254-96-6

ethyl (1S,5R,6S)-5-(1-ethylpropoxy)-7-oxabicyclo[4.1.0]hept-3-ene-3-carboxylate

726

2920 90 10

80841-78-7

4-(chloromethyl)-5-methyl-1,3-dioxol-2-one

436

2920 90 85

163133-43-5

4-(nitrooxy)butyl (2S)-2-(6-methoxy-2-naphthyl)propanoate

540

2921 49 80

259729-93-6

(1R)-1-[1-(4-chlorophenyl)cyclobutyl]-3-methylbutan-1-amine D-tartarate (1:1)

756

2921 49 80

3789-59-1

(1S)-1-phenylpropan-1-amine

559

2921 49 80

389056-74-0

(1S)-1-[1-(4-chlorophenyl)cyclobutyl]-3-methylbutan-1-amine D-tartarate (1:1)

558

2921 49 80

84467-54-9

1-[1-(4-chlorophenyl)cyclobutyl]-3-methylbutan-1-amine

480

2921 59 90

140-28-3

N, N'-dibenzylethane-1,2-diamine diacetate

226

2922 19 80

114247-09-5

(3R)-N-methyl-3-phenyl-3-[4-(trifluoromethyl)phenoxy]propan-1-amine hydrochloride

84

2922 19 80

115287-37-1

N-methyl-N-(4-nitrophenethyl)-2-(4-nitrophenoxy) ethan-1-amine

389

2922 19 80

168960-19-8

((1S,4R)-4-aminocyclopent-2-en-1-yl)methanol hydrochloride

669

2922 19 80

214353-17-0

1-(2-amino-5-chlorophenyl)-2,2,2-trifluoroethane-1,1-diol hydrochloride

42

2922 19 80

35320-23-1

(2R)-2-aminopropan-1-ol

512

2922 19 80

42142-52-9

3-(methylamino)-1-phenylpropan-1-ol

670

2922 19 80

467426-34-2

(2S)-2-(2-amino-5-chlorophenyl)-4-cyclopropyl-1,1,1-trifluorobut-3-yn-2-ol methanesulfonate (1:1.5)

547

2922 19 80

56796-66-8

4-(benzyloxy)-α1-[(tert-butylamino)methyl]benzene-1,3-dimethanol

575

2922 19 80

58997-87-8

2-(dimethylamino)-2-phenylbutan-1-ol

85

2922 29 00

115256-13-8

4-(1-{[2-(4-aminophenoxy)ethyl]methylamino}ethyl)aniline

552

2922 29 00

188690-84-8

(2S)-hydroxy(phenyl)acetic acid — (2R)-N-benzyl-1-(4-methoxyphenyl)propan-2-amine (1:1) (salt)

745

2922 29 00

202197-26-0

3-chloro-4-[(3-fluorobenzyl)oxy]aniline

471

2922 39 00

14189-82-3

(2E)-3-(N-methylanilino)acrylaldehyde

231

2922 49 95

209216-09-1

2-aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid hydrate

857

2922 49 95

223445-75-8

[(3S,4S)-1-(aminomethyl)-3,4-dimethylcyclopentyl]acetic acid

486

2922 49 95

26774-89-0

sodium 2-(cyclohexa-1,4-dien-1-yl)-2-[((E)-1-methoxy-1-oxobut-2-en-2-yl)amino]acetate

549

2922 50 00

174607-68-2

(1R)-1-[4-(benzyloxy)-3-(hydroxymethyl)phenyl]-2-(tert-butylamino)ethan-1-ol

48

2922 50 00

196810-09-0

methyl N-(2-benzoylphenyl)-L-tyrosinate

548

2922 50 00

50293-90-8

4-[(1R)-2-(tert-butylamino)-1-hydroxyethyl]-2-(hydroxymethyl)phenol hydrochloride

860

2922 50 00

62023-62-5

(2S,3S)-3-amino-2-hydroxy-4-phenylbutanoic acid

644

2922 50 00

653574-13-1

methyl N-(benzyloxycarbonyl)valyl-D-alloisoleucylthreonylnorvalinate

945

2922 50 00

71786-67-9

2-[benzyl(methyl)amino]-1-(3-hydroxyphenyl)ethan-1-one hydrochloride

18

2922 50 00

96072-82-1

1-[4-(benzyloxy)phenyl]-2-[(4-phenylbutan-2-yl)amino]propan-1-one

379

2923 20 00

4235-95-4

1,2-dioleoyl-sn-glycero-3-phosphocholine

377

2923 20 00

77286-66-9

2-O-methyl-1-O-octadecyl-sn-glycero-3-phosphocholine

198

2924 19 00

162537-11-3

N-(methoxycarbonyl)-3-methyl-L-valine

309

2924 19 00

186193-10-2

(2S)-2-{[3-(tert-butoxycarbonyl)-2,2-dimethylpropanoyl]oxy}-4-methylpentanoic acid

378

2924 19 00

228706-30-7

1,2-dioleoyl-sn-glycero-3-phospho[N-(4-carboxybutanoyl)ethanolamine]

12

2924 19 00

89182-60-5

1-deoxy-1-formamidohexitol

352

2924 29 95

132327-80-1

N2-[(9H-fluoren-9-ylmethoxy)carbonyl]-N5-trityl-L-glutamine

348

2924 29 95

132388-59-1

N2-[(9H-fluoren-9-ylmethoxy)carbonyl]-N4-trityl-L-asparagine

183

2924 29 95

170361-49-6

N-(3,4-dichlorophenyl)-N-{3-[(2,3-dihydroinden-2-yl)methylamino]propyl}-5,6,7,8-tetrahydronaphthalene-2-carboxamide

102

2924 29 95

194085-75-1

2-(2-chlorophenyl)-2-hydroxyethyl carbamate

398

2924 29 95

22871-58-5

3-amino-5-[(2-hydroxyethyl)carbamoyl]-2,4,6-triiodobenzoic acid

360

2924 29 95

244191-94-4

N-[(9H-fluoren-9-ylmethoxy)carbonyl]-α-L-glutamyl-N6-(tert-butoxycarbonyl)-L-lysyl-N-trityl-L-asparaginyl-α-L-glutamyl-N-trityl-L-glutaminyl-α-L-glutamyl-L-leucyl-L-leucyl-α-L-glutamyl-L-leucine, 1,4,6,9-tetra-tert-butyl ester

13

2924 29 95

28197-66-2

N-[3-acetyl-4-(oxiran-2-ylmethoxy)phenyl]butanamide

687

2924 29 95

325715-13-7

N-(3-acetylphenyl)-N-methylacetamide

347

2924 29 95

35661-39-3

N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-alanine

349

2924 29 95

35661-60-0

N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-leucine

598

2924 29 95

376348-76-4

ethyl (3S)-3-(4,4-difluorocyclohexane-1-carboxamido)-3-phenylpropanoate

599

2924 29 95

376348-77-5

4,4-difluoro-N-((1S)-3-hydroxy-1-phenylpropyl)cyclohexane-1-carboxamide

600

2924 29 95

376348-78-6

4,4-difluoro-N-((1S)-3-oxo-1-phenylpropyl)cyclohexane-1-carboxamide

619

2924 29 95

40371-50-4

(2S)-4-{[(benzyloxy)carbonyl]amino}-2-hydroxybutanoic acid

731

2924 29 95

481659-97-6

tert-butyl {(1S)-2-[benzyl(methyl)amino]-2-oxo-1-phenylethyl}carbamate hydrochloride

411

2924 29 95

49705-98-8

benzyl ((1S,2R)-1-carbamoyl-2-hydroxypropyl)carbamate

144

2924 29 95

53947-84-5

2-(carboxyacetamido)benzoic acid

487

2924 29 95

6485-67-2

(2R)-2-amino-2-phenylacetamide

371

2924 29 95

65864-22-4

L-phenylalaninamide

696

2924 29 95

667937-05-5

3-[4-(trifluoromethyl)anilino]pentanamide

350

2924 29 95

71989-14-5

4-tert-butyl N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-aspartate

351

2924 29 95

71989-18-9

5-tert-butyl N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-glutamate

353

2924 29 95

71989-20-3

N2-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-glutamine

355

2924 29 95

71989-23-6

N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-isoleucine

356

2924 29 95

71989-26-9

N6-(tert-butoxycarbonyl)-N2-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-lysine

367

2924 29 95

71989-33-8

O-tert-butyl-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-serine

368

2924 29 95

71989-35-0

O-tert-butyl-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-threonine

370

2924 29 95

71989-38-3

O-tert-butyl-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-tyrosine

412

2924 29 95

80082-51-5

3-amino-2-{[(benzyloxy)carbonyl]amino}-1-methyl-3-oxopropyl methanesulfonate

197

2924 29 95

98760-08-8

tert-butyl [1-((2S)-oxiran-2-yl)-2-phenylethyl]carbamate

317

2925 29 00

249561-98-6

tris{[(2Z)-2-chloro-3-(dimethylamino)prop-2-en-1-ylidene]dimethylammonium}

hexafluorophosphate(3-)

215

2925 29 00

3382-63-6

4-{(E)-[(4-fluorophenyl)imino]methyl}phenol

938

2926 90 95

114772-54-2

4'-(bromomethyl)biphenyl-2-carbonitrile

142

2926 90 95

152630-47-2

1-[3-(cyclopentyloxy)-4-methoxyphenyl]-4-oxocyclohexane-1-carbonitrile

143

2926 90 95

152630-48-3

dimethyl 4-cyano-4-[3-(cyclopentyloxy)-4-methoxyphenyl]heptanedioate

585

2926 90 95

192869-10-6

2-iodo-3,4-dimethoxy-6-nitrobenzonitrile

586

2926 90 95

192869-24-2

6-amino-2-iodo-3,4-dimethoxybenzonitrile

539

2926 90 95

28049-61-8

1-(4-chlorophenyl)cyclobutane-1-carbonitrile

528

2926 90 95

31915-40-9

N-[1-cyano-2-(4-hydroxyphenyl)-1-methylethyl]acetamide

673

2926 90 95

474645-97-1

(3R)-3-aminopentanenitrile methanesulfonate

803

2926 90 95

604784-44-3

tert-butylammonium (Z)-3-cyano-5-methylhex-3-enoate

287

2928 00 90

212631-79-3

2-(2-chloro-4-iodoanilino)-N-(cyclopropylmethoxy)-3,4-difluorobenzamide

33

2928 00 90

253605-31-1

N-hydroxy-2-methylpropan-2-amine acetate (salt) or tert-butylhydroxylamine acetate (salt)

49

2928 00 90

618-26-8

1-methyl-1-phenylhydrazine sulfate (2:1)

403

2929 90 00

204254-98-8

ethyl (3R,4S,5R)-5-azido-3-(1-ethylpropoxy)-4-hydroxycyclohex-1-ene-1-carboxylate

405

2929 90 00

204255-06-1

ethyl (3R,4R,5S)-4-acetamido-5-azido-3-(1-ethylpropoxy)cyclohex-1-ene-1-carboxylate

748

2930 90 85

104458-24-4

2-mesylethan-1-amine hydrochloride

399

2930 90 85

153277-33-9

methyl N-[(benzyloxy)carbonyl]-S-phenyl-L-cysteinate

862

2930 90 85

15570-12-4

3-methoxybenzene-1-thiol

56

2930 90 85

16188-55-9

[4-(methylsulfanyl)phenyl]acetic acid

26

2930 90 85

225652-11-9

1-(4-chlorophenoxy)-4-(methylsulfanyl)benzene or 4-chlorophenyl 4-(methylsulfanyl)phenyl ether

339

2930 90 85

2736-23-4

2,4-dichloro-5-mesylbenzoic acid

595

2930 90 85

289717-37-9

N, N-dimethyl-2-[4-(methylsulfanyl)phenoxy]benzylamine hydrochloride

742

2930 90 85

346413-00-1

1-(4-ethoxyphenyl)-2-(4-mesylphenyl)ethan-1-one

358

2930 90 85

3483-12-3

(2R,3S)-1,4-disulfanylbutane-2,3-diol or dithiothreitol

594

2930 90 85

364323-64-8

2-[4-(methylsulfanyl)phenoxy]benzaldehyde

864

2930 90 85

40248-84-8

3-sulfanylphenol

324

2930 90 85

50413-24-6

2-bromo-1-(4-mesylphenyl)ethan-1-one

65

2930 90 85

90536-66-6

(4-mesylphenyl)acetic acid

206

2931 00 95

123599-82-6

{[2-methyl-1-(propionyloxy)propoxy](4-phenylbutyl)phosphoryl}acetic acid

58

2931 00 95

27784-76-5

tert-butyl (diethoxyphosphoryl)acetate

789

2931 00 95

649761-22-8

(1R,5S)-5-[dimethyl(phenyl)silyl]-2-(hydroxymethyl)cyclopent-2-ene-1-carboxylic acid — (1R,2R)-2-amino-1-(4-nitrophenyl)propane-1,3-diol (1:1) (salt)

391

2931 00 95

86552-32-1

(4-phenylbutyl)phosphinic acid

747

2932 19 00

27329-70-0

(5-formyl-2-furyl)boronic acid

762

2932 19 00

37076-71-4

1,2,3-tri-O-acetyl-5-deoxy-D-ribofuranose

700

2932 19 00

87392-07-2

(2S)-tetrahydrofuran-2-carboxylic acid

582

2932 29 85

122111-01-7

[(2R)-2-(benzoyloxy)-4,4-difluoro-5-oxotetrahydrofuran-2-yl]methyl benzoate

78

2932 29 85

142680-85-1

(25S)-25-cyclohexyl-25-de(sec-butyl)-5-O-demethyl-22,23-dihydroavermectin A1a

244

2932 29 85

145667-75-0

(3aR,4R,5R,6aS)-5-hydroxy-4-((3R)-3-hydroxy-5-phenylpentyl)hexahydrocyclopenta[b]furan-2-one

79

2932 29 85

220119-16-4

(25S)-cyclohexyl-25-de(sec-butyl)- 5-demethoxy-5-oxo-22,23-dihydroavermectin A1a

942

2932 29 85

221129-55-1

(6R)-4-hydroxy-6-phenethyl-6-propyl-5,6-dihydro-2H-pyran-2-one

115

2932 29 85

51559-36-5

5-methoxy-2H-chromen-2-one

660

2932 29 85

95716-70-4

7α-(methoxycarbonyl)-3-oxo-17α-pregna-4,9(11)-diene-21,17-carbolactone

703

2932 29 85

96829-59-3

(1S,3E,6E)-1-[((2S,3S)-3-hexyl-4-oxooxetan-2-yl)methyl]dodeca-3,6-dien-1-yl N-formyl-L-leucinate

37

2932 99 70

124655-09-0

tert-butyl [(4R,6S)-6-(hydroxymethyl)-2,2-dimethyl-1,3-dioxan-4-yl]acetate

567

2932 99 70

130064-21-0

1-{2-hydroxy-4-[(tetrahydropyran-2-yl)oxy]phenyl}-2-{4-[(tetrahydropyran-2-yl)oxy]phenyl}ethan-1-one

156

2932 99 70

167256-05-5

methyl (1S,2S)-1-(1,3-benzodioxol-5-yl)-3-(2-hydroxy-4-methoxyphenyl)-5-propoxyindane-2-carboxylate

157

2932 99 70

191106-49-7

methyl (1S,2S)-1-(1,3-benzodioxol-5-yl)-3-[2-(benzyloxy)-4-methoxyphenyl]-5-propoxyindane-2-carboxylate

189

2932 99 70

192201-93-7

2-({3-[5-(6-methoxy-1-naphthyl)-1,3-dioxan-2-yl]propyl}methylamino)-N-methylacetamide

127

2932 99 70

196303-01-2

(7S)-7-methyl-5-(4-nitrophenyl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]isochromene

62

2932 99 70

7772-94-3

2-acetamido-2-deoxy-β-D-mannopyranose

607

2932 99 85

115437-18-8

(2α,4α,5β,7β,10β,13β)-4-acetoxy-1,10,13-trihydroxy-9-oxo-7-[(triethylsilyl)oxy]-5,20-epoxytax-11-en-2-yl benzoate

608

2932 99 85

115437-21-3

(4α)-4,10-diacetoxy-1,13-dihydroxy-9-oxo-7-[(triethylsilyl)oxy]-5,20-epoxytax-11-en-2-yl benzoate

54

2932 99 85

130525-58-5

methyl 5-acetamido-7,8,9-O-triacetyl-2,6-anhydro-4-azido-3,4,5-trideoxy-D-glycero-D-galacto-non-2-enonate

609

2932 99 85

149107-93-7

(2α,4α,5β,7β,10β,13α)-4,10-diacetoxy-13-{[(2R,3S)-3-benzamido-2-(1-methoxy-1-methylethoxy)-3-phenylpropanoyl]oxy}-1-hydroxy-9-oxo-7-[(triethylsilyl)oxy]-5,20-epoxytax-11-en-2-yl benzoate

652

2932 99 85

199796-52-6

(2α,4α,7β,10β,13α)-4,10-diacetoxy-13-({(2R,3S)-3-benzamido-2-[((4Z,7Z,10Z,13Z,16Z,19Z)-docosa-4,7,10,13,16,19-hexaenoyl)oxy]-3-phenylpropanoyl}oxy)-1,7-dihydroxy-9-oxo-5,20-epoxytax-11-en-2-yl benzoate

11

2932 99 85

65293-32-5

N-β-D-glucopyranosylformamide

590

2933 19 90

334828-10-3

4-amino-5-ethyl-1-(2-methoxyethyl)pyrazole-3-carboxamide

511

2933 21 00

186462-71-5

(1R,2R,5S,6R)-2',5'-dioxospiro[bicyclo[3.1.0]hexane-2,4'-imidazolidine]-6-carboxylic acid

354

2933 29 90

109425-51-6

N2-[(9H-fluoren-9-ylmethoxy)carbonyl]-N-trityl-L-histidine

263

2933 29 90

178982-67-7

2-[(benzyloxy)methyl]-4-isopropylimidazole

359

2933 29 90

244191-88-6

N-acetyl-O-tert-butyl-L-tyrosyl-O-tert-butyl-L-threonyl-O-tert-butyl-L-seryl-L-leucyl-L-isoleucyl-N1-trityl-L-histidyl-O-tert-butyl-L-seryl-L-leucyl-L-isoleucyl-α-L-glutamyl-α-L-glutamyl-O-tert-butyl-L-seryl-N-trityl-L-glutaminyl-N-trityl-L-asparaginyl-N-trityl-L-glutaminyl-L-glutamine, 10,11-di-tert-butyl ester

365

2933 29 90

244244-26-6

N-acetyl-O-tert-butyl-L-tyrosyl-O-tert-butyl-L-threonyl-O-tert-butyl-L-seryl-L-leucyl-L-isoleucyl-N1- trityl-L-histidyl-O-tert-butyl-L-seryl-L-leucyl-L-isoleucyl-α-L-glutamyl-α-L-glutamyl-O-tert-butyl-L-seryl-N-trityl-L-glutaminyl-N-trityl-L-asparaginyl-N-trityl-L-glutaminyl-L-glutaminyl-α-L-glutamyl-N6-(tert-butoxycarbonyl)-L-lysyl-N-trityl-L-asparaginyl-α-L-glutamyl-N-trityl-L-glutaminyl-α-L-glutamyl-L-leucyl-L-leucyl-α-L-glutamyl-L-leucyl-α-L-aspartyl-N6-(tert-butoxycarbonyl)-L-lysyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-alanyl-O-tert-butyl-L-seryl-L-leucyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-N-trityl-L-asparaginyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-phenylalaninamide, hepta-tert-butyl ester

583

2933 29 90

68283-19-2

(2-butylimidazol-5-yl)methanol

954

2933 39 99

0-00-0

11-ethyl-5-methyl-8-{2-[(1-oxo-1λ4-quinolin-4-yl)oxy]ethyl}-11H-dipyrido[3,2-b:2',3'-e][1,4]diazepin-6(5H)-one

119

2933 39 99

100238-42-4

4-(2-piperidin-1-ylethoxy)phenol

541

2933 39 99

103129-82-4

3-ethyl 5-methyl 2-[(2-aminoethoxy)methyl]-4-(2-chlorophenyl)-6-methyl-1,4-dihydropyridine-3,5-dicarboxylate

167

2933 39 99

127293-57-6

(1R)-1-(4-chlorophenyl)-2-[4-(4-fluorobenzyl)piperidin-1-yl]ethan-1-ol

16

2933 39 99

158878-47-8

(3R,5R)-3-{(E)-2-[4-(4-fluorophenyl)-2,6-diisopropyl-5-(methoxymethyl)pyridin-3-yl]vinyl}-5-hydroxycyclohexan-1-one

14

2933 39 99

159813-78-2

(3R,5S,6E)-7-[4-(4-fluorophenyl)-2,6-diisopropyl-5-(methoxymethyl)pyridin-3-yl]-3,5-dihydroxyhept-6-enoic acid

621a

2933 39 99

161417-03-4

2-methyl-3-((2S)-pyrrolidin-2-ylmethoxy)pyridine

9

2933 39 99

177964-68-0

3-[4-(4-fluorophenyl)-2,6-diisopropyl-5-(methoxymethyl)pyridin-3-yl]acrylaldehyde

168

2933 39 99

178460-82-7

(1R)-1-(4-chlorophenyl)-2-[4-(4-fluorobenzyl)piperidin-1-yl]ethan-1-ol hydrochloride

264

2933 39 99

178981-89-0

{5-[(3,5-dichlorophenyl)sulfanyl]-4-isopropyl-1-(pyridin-4-ylmethyl)imidazol-2-yl}methanol

173

2933 39 99

188396-54-5

1-(2-biphenyl-4-ylethyl)-4-[3-(trifluoromethyl)phenyl]-1,2,3,6-tetrahydropyridine hydrochloride

875

2933 39 99

19395-39-2

2-phenyl-2-piperidin-2-ylacetamide

196

2933 39 99

198904-85-7

tert-butyl 2-(4-pyridin-2-ylbenzyl)hydrazine-1-carboxylate

199

2933 39 99

198904-86-8

tert-butyl 2-{(2S,3S)-3-[(tert-butoxycarbonyl)amino]-2-hydroxy-4-phenylbutyl}-2-[4-(pyridin-2-yl)benzyl]hydrazine-1-carboxylate

840

2933 39 99

213839-64-6

N-{2-[5-(aminoiminomethyl)-2-hydroxyphenoxy]-3,5-difluoro-6-[3-(1-methyl-4,5-dihydroimidazol-2-yl)phenoxy]pyridin-4-yl]-N-methyglycine dihydrochloride

442

2933 39 99

221180-26-3

4-amino-5-chloro-2-methoxy-N-(3-methoxypiperidin-4-yl)benzamide

318

2933 39 99

221615-75-4

2-(4-mesylphenyl)-1-(6-methylpyridin-3-yl)- ethan-1-one

690

2933 39 99

230615-52-8

2,3,4,5-tetrahydro-1H-1,5-methano-3-benzazepine hydrochloride

661

2933 39 99

230615-59-5

7,8-dinitro-3-(trifluoroacetyl)-2,3,4,5-tetrahydro-1H-1,5-methano-3-benzazepine

765

2933 39 99

25333-42-0

(3R)-quinuclidin-3-ol

565

2933 39 99

26815-04-3

4-(2-piperidin-1-ylethoxy)benzaldehyde

842

2933 39 99

280129-82-0

4-({2-[(benzyloxy)methyl]-4-isopropylimidazol-1-yl}methyl)pyridine oxalate (1:2)

490

2933 39 99

319460-85-0

N-methyl-2-{[3-((E)-2-pyridin-2-ylvinyl)-1H-indazol-6-yl]sulfanyl}benzamide

489

2933 39 99

319460-94-1

N-(2-fluoro-5-{[3-((E)-2-pyridin-2-ylvinyl)-1H-indazol-6-yl]amino}phenyl)-1,3-dimethylpyrazole-5-carboxamide

579

2933 39 99

37699-43-7

2,3-dimethyl-4-nitropyridine 1-oxide

210

2933 39 99

4021-07-2

3-methylpyridine-2-carboxylic acid

649

2933 39 99

423165-13-3

8-benzyl-3-exo-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)-8-azabicyclo[3.2.1]octane

951

2933 39 99

429659-01-8

ethyl N-[4-(methylamino)-3-nitrobenzoyl]-N-pyridin-2-yl-ß-alaninate

560

2933 39 99

43200-82-4

6-(5-chloropyridin-2-yl)-5H-pyrrolo[3,4-b]pyrazine-5,7(6H)-dione

564

2933 39 99

440634-25-3

tert-butyl 4-{2-[4-(mesyloxy)piperidin-1-yl]-2-oxoethyl}piperidine-1-carboxylate

538

2933 39 99

58859-46-4

ethyl 4-aminopiperidine-1-carboxylate

626

2933 39 99

78750-68-2

4-[(3-aminopyridin-2-yl)amino]phenol

513

2933 39 99

84449-81-0

4-(2-piperidin-1-ylethoxy)benzoyl chloride hydrochloride

948

2933 49 90

0-00-0

2-(ethylamino)-5-[2-(quinolin-4-yloxy)ethyl]nicotinic acid

483

2933 49 90

10500-57-9

5,6,7,8-tetrahydroquinoline

149

2933 49 90

106635-86-3

2,6-dimethoxy-4-methyl-5-[3-(trifluoromethyl)phenoxy]quinolin-8-amine

647

2933 49 90

118864-75-8

(1S)-1-phenyl-1,2,3,4-tetrahydroisoquinoline

36

2933 49 90

172649-40-0

3-[(4S)-5-oxo-2-(trifluoromethyl)-1,4,5,6,7,8-hexahydroquinolin-4-yl]benzonitrile

623

2933 49 90

189279-58-1

1-(6-amino-3,5-difluoropyridin-2-yl)-8-chloro-6-fluoro-7-(3-hydroxyazetidin-1-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylic acid

150

2933 49 90

189746-15-4

2,6-dimethoxy-4-methyl-8-nitro-5-[3-(trifluoromethyl)phenoxy]quinoline

152

2933 49 90

189746-19-8

5-chloro-2,6-dimethoxy-4-methylquinoline

151

2933 49 90

189746-21-2

5-chloro-2,6-dimethoxy-4-methyl-8-nitroquinoline

434

2933 49 90

194804-45-0

ethyl 1-cyclopropyl-8-(difluoromethoxy)-7-((1R)-1-methyl-2-tritylisoindolin-5-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylate

433

2933 49 90

194805-07-7

ethyl 7-bromo-1-cyclopropyl-8-(difluoromethoxy)-4-oxo-1,4-dihydroquinoline-3-carboxylate

705A

2933 49 90

209909-03-5

(2-chloro-6,7-difluoroquinolin-3-yl)methanol

704A

2933 49 90

220998-08-3

{2,7-dichloro-6-methyl-4-[(4-methylpiperidin-1-yl)methyl]quinolin-3-yl}methanol

386

2933 49 90

287930-77-2

(1S)-1-{3-[(E)-2-(7-chloroquinolin-2-yl)vinyl]phenyl}-3-[2-(1-hydroxy-1-methylethyl)phenyl]propan-1-ol

387

2933 49 90

287930-78-3

methyl 2-((3S)-3-{3-[(E)-2-(7-chloroquinolin-2-yl)vinyl]phenyl}-3-hydroxypropyl)benzoate hydrate

674

2933 49 90

474645-93-7

methyl [2-ethyl-6-(trifluoromethyl)-1,2,3,4-tetrahydroquinolin-4-yl]carbamate

153

2933 49 90

6340-55-2

2,6-dimethoxy-4-methylquinoline

664

2933 49 90

79276-06-5

tert-butyl (3S)-1,2,3,4-tetrahydroisoquinoline-3-carboxylate 4-methylbenzenesulfonate

455

2933 59 95

119532-26-2

1-(2,3-dichlorophenyl)piperazine

80

2933 59 95

137234-74-3

4-chloro-6-ethyl-5-fluoropyrimidine

509

2933 59 95

137281-39-1

4-[2-(2-amino-4-oxo-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-5-yl)ethyl]benzoic acid

39

2933 59 95

140373-09-7

4-{[(3-{[(2,2-dimethylpropanoyl)oxy]methyl}-2,7-dimethyl-4-oxo-3,4-dihydroquinazolin-6-yl)methyl](prop-2-yn-1-yl)amino}-2-fluorobenzoic acid

531

2933 59 95

14080-23-0

pyrimidine-2-carbonitrile

38

2933 59 95

160009-37-0

methyl 4-(4-fluorophenyl)-6-isopropyl-2-(N-methylmethanesulfonamido)]pyrimidine-5-carboxylate

744

2933 59 95

16064-08-7

6-iodoquinazolin-4(1H)-one

123

2933 59 95

167465-36-3

(2R)-1-[4-((1aR,10bS)-1,1-difluoro-1,1a,6,10b-tetrahydrodibenzo[a, e]cyclopropa[c][7]annulen-6-yl)piperazin-1-yl]-3-[(quinolin-5-yl)oxy]propan-2-ol trihydrochloride

73

2933 59 95

188416-20-8

3-(6-chloro-5-fluoropyrimidin-4-yl)-2-(2,4-difluorophenyl)-1-(1H-1,2,4-triazol-1-yl)butan-2-ol hydrochloride

81

2933 59 95

188416-28-6

4-(1-bromoethyl)-6-chloro-5-fluoropyrimidine

112

2933 59 95

192725-50-1

(2S)-3-methyl-2-(2-oxohexahydropyrimidin-1-yl)butanoic acid

133

2933 59 95

192726-06-0

(2S)-N-[(1S,3S,4S)-4-amino-1-benzyl-3-hydroxy-5-phenylpentyl]-3-methyl-2-(2-oxotetrahydropyrimidin-1(2H)-yl)butanamide — 5-oxopyrrolidine-2-carboxylic acid (1:1) (salt)

790

2933 59 95

19916-73-5

6-(benzyloxy)-9H-purin-2-amine

261

2933 59 95

214287-88-4

(4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluoromethyl)-3,4-dihydroquinazolin-2(1H)-one

259

2933 59 95

214287-99-7

(4S)-6-chloro-4-((E)-2-cyclopropylvinyl)-4-(trifluoromethyl)-3,4-dihydroquinazolin-2(1H)-one

653

2933 59 95

225916-82-5

8-chloro-5-((4Z,7Z,10Z,13Z,16Z,19Z)-docosa-4,7,10,13,16,19-hexaenoyl)-11-(4-methylpiperazin-1-yl)-5H-dibenzo[b, e][1,4]diazepine

746

2933 59 95

231278-20-9

N-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-iodoquinazolin-4-amine

256

2933 59 95

247565-04-4

(4S)-6-chloro-4-(cyclopropylethynyl)-3-((R)-1-phenylethyl)-4-(trifluoromethyl)-3,4-dihydroquinazolin-2(1H)-one

554

2933 59 95

345217-02-9

1-[(1S,2S)-2-(benzyloxy)-1-ethylpropyl]-N-{4-[4-(4-hydroxyphenyl)piperazin-1-yl]phenyl}hydrazine-1-carboxamide

313

2933 59 95

487-21-8

pteridine-2,4(1H,3H)-dione

958

2933 59 95

518048-03-8

2-(1-amino-1-methylethyl)-N-(4-fluorobenzyl)-5-hydroxy-1-methyl-6-oxo-1,6-dihydropyrimidine-4-carboxamide

949

2933 59 95

57061-71-9

1-(2-chloroethyl)-4-[3-(trifluoromethyl)phenyl]piperazine dihydrochloride

561

2933 59 95

59878-63-6

6-(5-chloropyridin-2-yl)-7-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyrazin-5-yl piperazine-1-carboxylate

830

2933 59 95

599179-03-0

1-(4,6-dimethylpyrimidine-5-carbonyl)-

4-((3S)-4-{(1R)-2-methoxy-1-[4-(trifluoromethyl)phenyl]ethyl}-3-methylpiperazin-1-yl)-4-methylpiperidine maleate (1:1)

828

2933 59 95

612494-10-7

1-{(1R)-2-methoxy-1-[4-(trifluoromethyl)phenyl]ethyl}-2-methylpiperazine D-tartarate (1:1)

829

2933 59 95

612543-01-8

1-(4,6-dimethylpyrimidine-5-carbonyl)piperidin-4-one

791

2933 59 95

649761-23-9

(1S,2S,3S,5S)-5-[2-amino-6-(benzyloxy)-9H-purin-9-yl]-2-[(benzyloxy)methyl]-3-[dimethyl(phenyl)silyl]-1-(hydroxymethyl)cyclopentan-1-ol

792

2933 59 95

649761-24-0

2-amino-9-{(1S,3R,4S)-3-[(benzyloxy)methyl]-4-[dimethyl(phenyl)silyl]-2-methylidenecyclopentyl}-9H-purin-6(1H)-one

835

2933 59 95

654671-77-9

(2R)-4-oxo-4-[3-(trifluoromethyl)-5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-1-(2,4,5-trifluorophenyl)butan-2-amine phosphate (1:1) hydrate

946

2933 59 95

7139-02-8

2,6-dichloro-4,8-dipiperidinopyrimido[5,4-d]pyrimidine

457

2933 79 00

105318-28-3

((2S,3S)-2-{(1R)-2-[(4-chlorophenyl)sulfanyl]-1-methyl-2-oxoethyl}-3-((1R)-1-hydroxyethyl)-4-oxoazetidin-1-yl)acetic acid

610

2933 79 00

133066-59-8

(3R,4S)-2-oxo-4-phenylazetidin-3-yl acetate

60

2933 79 00

148776-18-5

(2-oxo-1-phenylpyrrolidin-3-yl)triphenylphosphonium bromide

612

2933 79 00

149107-92-6

1-benzoyl-3-(1-methoxy-1-methylethoxy)-4-phenylazetidin-2-one

692

2933 79 00

162142-14-5

1-cyclopentyl-3-ethyl-1,4,5,6-tetrahydro-7H-pyrazolo[3,4-c]pyridin-7-one

50

2933 79 00

198213-15-9

sodium 3-(methoxycarbonyl)-2-oxo-1,2,5,6-tetrahydropyridin-4-olate

188

2933 79 00

205881-86-3

6-fluoro-9-methyl-2-phenyl-4-(pyrrolidine-1-carbonyl)-9H-pyrido[3,4-b]indol-1(2H)-one

176

2933 79 00

244080-24-8

1-ethyl-9-methoxy-2,6,7,12-tetrahydroindolo[2,3-a]quinolizin-4(3H)-one

491

2933 79 00

283173-50-2

8-fluoro-2-{4-[(methylamino)methyl]phenyl}-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-one

693

2933 79 00

303752-13-8

1-cyclopentyl-3-ethyl-6-(4-methoxybenzyl)-1,4,5,6-tetrahydro-7H-pyrazolo[3,4-c]pyridin-7-one 4-methylbenzene-1-sulfonate

148

2933 79 00

3197-25-9

2-(4-oxopentyl)-1H-isoindole-1,3(2H)-dione

776

2933 79 00

341031-54-7

N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fluoro-2-oxo-1,2-dihydro-3H-indol-3-ylidene)methyl]-2,4-dimethylpyrrole-3-carboxamide L-malate (1:1)

713

2933 79 00

43200-81-3

6-(5-chloropyridin-2-yl)-7-hydroxy-6,7-dihydro-5H-pyrrolo[3,4-b]pyrazin-5-one

154

2933 79 00

5342-23-4

6-methoxy-4-methylquinolin-2(1H)-one

413

2933 79 00

80082-62-8

tetrabutylammonium (2S,3S)-3-{[(benzyloxy)carbonyl]amino}-2-methyl-4-oxoazetidine-1-sulfonate

414

2933 79 00

80082-65-1

(2S,3S)-3-amino-2-methyl-4-oxoazetidine-1-sulfonic acid

140

2933 99 40

193077-87-1

[(2S)-7-(2-methoxy-2-oxoethyl)-4-methyl-3-oxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-2-yl]acetic acid

139

2933 99 40

210288-67-8

[(2S)-7-iodo-4-methyl-3-oxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-2-yl]acetic acid

392

2933 99 90

103201-78-1

4-cyclohexylproline

120

2933 99 90

113963-68-1

3,4-di(indol-3-yl)-1-methylpyrrole-2,5-dione

322

2933 99 90

119192-10-8

4-[(1H-1,2,4-triazol-1-yl)methyl]aniline

422

2933 99 90

120807-02-5

(4S)-N-benzoyl-4-(mesyloxy)-L-proline

369

2933 99 90

143824-78-6

N1-(tert-butoxycarbonyl)-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-tryptophan

227

2933 99 90

14907-27-8

methyl D-tryptophanate hydrochloride

4

2933 99 90

149365-59-3

dibenzyl 5,5'-[(3,4-diethylpyrrole-2,5-diyl)bis(methylene)]bis[4-(3-methoxy-3-oxopropyl)-3-methylpyrrole-2-carboxylate]

5

2933 99 90

149365-62-8

5,5'-[(3,4-diethylpyrrole-2,5-diyl)bis(methylene)]bis[4-(3-hydroxypropyl)-3-methylpyrrole-2-carbaldehyde]

940

2933 99 90

152628-02-9

1,4'-dimethyl-2'-propyl-1H,1'H-2,6'-bibenzimidazole

939

2933 99 90

152628-03-0

4-Methyl-2-propylbenzimidazole-6-carboxylic acid

323

2933 99 90

160194-39-8

2-{5-[(1H-1,2,4-triazol-1-yl)methyl]indol-3-yl}ethan-1-ol

312

2933 99 90

16298-03-6

methyl 3-aminopyrazine-2-carboxylate

35

2933 99 90

171964-73-1

[N-(4-methoxybenzoyl)-L-valyl]-N-[(1S)-3,3,3-trifluoro-1-isopropyl-2-oxopropyl]-L-prolinamide

230

2933 99 90

172733-42-5

sodium [(1-benzyl-2-ethyl-3-oxamoylindol-4-yl)oxy]acetate

87

2933 99 90

180637-89-2

3-[((2R)-1-methylpyrrolidin-2-yl)methyl]-5-[(E)-2-(phenylsulfonyl)vinyl]indole

677

2933 99 90

180915-94-0

1-{2-[4-(6-methoxy-3,4-dihydro-1-naphthyl)phenoxy]ethyl}pyrrolidine

676

2933 99 90

180915-95-1

1-{2-[4-(2-bromo-6-methoxy-3,4-dihydro-1-naphthyl)phenoxy]ethyl}pyrrolidine

31

2933 99 90

181827-47-4

[N-(methoxycarbonyl)-L-valyl]-L-proline

86

2933 99 90

188113-71-5

1-acetyl-3-[((2R)-1-methylpyrrolidin-2-yl)methyl]-5-[(E)-2-(phenylsulfonyl)vinyl]indole

27

2933 99 90

193274-37-2

3a-benzyl-2-methyl-2,3a,4,5,6,7-hexahydro-3H-pyrazolo[4,3-c]pyridin-3-one L-tartarate

137

2933 99 90

197143-35-4

(3Z)-4-(aminomethyl)pyrrolidin-3-one O-methyloxime dihydrochloride

404

2933 99 90

204255-02-7

ethyl (1R,5R,6R)-5-(1-ethylpropoxy)-7-azabicyclo[4.1.0]hept-3-ene-3-carboxylate

794

2933 99 90

210558-66-0

(1R,2S)-1-phenyl-2-pyrrolidin-1-ylpropan-1-ol hydrochloride

319

2933 99 90

219909-83-8

3-((4S)-4-sulfanyl-L-prolinamidol)benzoic acid hydrochloride

634

2933 99 90

221030-56-4

2-(4-fluorophenyl)-4-(3-hydroxy-3-methylbutoxy)-5-(4-mesylphenyl)pyridazin-3(2H)-one

743

2933 99 90

221148-46-5

2-(4-ethoxyphenyl)-3-(4-mesylphenyl)pyrazolo[1,5-b]pyridazine

245

2933 99 90

227025-33-4

1-benzyl-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one

441

2933 99 90

235106-62-4

2,2'-[(4-hydroxyphenyl)methylene]bis(4-{(E)-[(5-methyl-1H-tetrazol-1-yl)imino]methyl}phenol)

362

2933 99 90

244191-95-5

α-L-aspartyl-N6-(tert-butoxycarbonyl)-L-lysyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-alanyl-O-tert-butyl-L-seryl-L-leucyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-N-trityl-L-asparaginyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-phenylalaninamide, tert-butyl ester

361

2933 99 90

244191-96-6

N-[(9H-fluoren-9-ylmethoxy)carbonyl]-α-L-aspartyl-N6-(tert-butoxycarbonyl)-L-lysyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-alanyl-O-tert-butyl-L-seryl-L-leucyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-N-trityl-L-asparaginyl-N1-(tert-butoxycarbonyl)-L-tryptophan, 1-tert-butyl ester

363

2933 99 90

244244-29-9

N-[(9H-fluoren-9-ylmethoxy)carbonyl]-α-L-glutamyl-N6-(tert-butoxycarbonyl)-L-lysyl-N-trityl-L-asparaginyl-α-L-glutamyl-N-trityl-L-glutaminyl-α-L-glutamyl-L-leucyl-L-leucyl-α-L-glutamyl-L-leucyl-α-L-aspartyl-N6-(tert-butoxycarbonyl)-L-lysyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-alanyl-O-tert-butyl-L-seryl-L-leucyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-N-trityl-L-asparaginyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-phenylalaninamide, penta-tert-butyl ester

364

2933 99 90

244244-31-3

α-L-glutamyl-N6-(tert-butoxycarbonyl)-L-lysyl-N-trityl-L-asparaginyl-α-L-glutamyl-N-trityl-L-glutaminyl-α-L-glutamyl-L-leucyl-L-leucyl-α-L-glutamyl-L-leucyl-α-L-aspartyl-N6-(tert-butoxycarbonyl)-L-lysyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-alanyl-O-tert-butyl-L-seryl-L-leucyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-N-trityl-L-asparaginyl-N1-(tert-butoxycarbonyl)-L-tryptophyl-L-phenylalaninamide, penta-tert-butyl ester monohydrochloride

646

2933 99 90

251579-55-2

(N-acetyl-N-methylglycyl)glycylvalyl-D-alloisoleucylthreonylnorvalylisoleucylarginyl(N-ethylprolinamide) monoacetate (salt)

581

2933 99 90

252742-72-6

5-(chloromethyl)-1,2-dihydro-3H-1,2,4-triazol-3-one

246

2933 99 90

269731-84-2

(5R,6R)-1-benzyl-5-hydroxy-6-(methylamino)-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one

563

2933 99 90

272107-22-9

3,10-dibromo-8-chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridine

420

2933 99 90

31560-19-7

N-benzoyl-4-hydroxyproline

421

2933 99 90

31560-20-0

methyl N-benzoyl-4-hydroxyprolinate

91

2933 99 90

32065-66-0

2-(dimethoxymethyl)quinoxaline 1,4-dioxide

741

2933 99 90

346412-97-3

1-aminopyridazinium hexafluorophosphate(1-)

373

2933 99 90

39968-33-7

3H-[1,2,3]triazolo[4,5-b]pyridin-3-ol

645

2933 99 90

442526-89-8

isoleucylarginyl(N-ethylprolinamide) dihydrochloride

729

2933 99 90

481659-93-2

ethyl 1-methyl-5-[4'-(trifluoromethyl)biphenyl-2-carboxamido]indole-2-carboxylate

730

2933 99 90

481659-96-5

potassium 1-methyl-5-[4'-(trifluoromethyl)biphenyl-2-carboxamido]indole-2-carboxylate

311

2933 99 90

5424-01-1

3-aminopyrazine-2-carboxylic acid

724

2933 99 90

61607-68-9

1-[2-(dimethylamino)ethyl]-4,5-dihydro-1H-tetrazole-5-thione

488

2933 99 90

62893-24-7

(6-ethyl-4,5-dioxohexahydropyridazine-3-carboxamido)(4-hydroxyphenyl)acetic acid

223

2933 99 90

6548-09-0

5-bromotryptophan

728

2933 99 90

71056-57-0

ethyl 1-methyl-5-nitroindole-2-carboxylate

19

2933 99 90

75302-98-6

2-tert-butoxy-2-oxoethyl [1-(4-chlorobenzoyl)-5-methoxy-2-methylindol-3-yl]acetate

537

2933 99 90

84946-20-3

2-chloro-1-(4-fluorobenzyl)benzimidazole hydrochloride

72

2933 99 90

86404-63-9

1-(2,4-difluorophenyl)-2-(1H-1,2,4-triazol-1-yl)ethan-1-one

396

2933 99 90

92992-17-1

1-(methoxycarbonyl)-2,3-dihydro-1H-pyrrolizine-7-carboxylic acid

416

2933 99 90

96314-26-0

(4S)-4-phenyl-L-proline

737

2934 10 00

115065-79-7

(2E)-2-(2-{[(benzyloxy)carbonyl]amino}-1,3-thiazol-4-yl)-5-[(3-methylbut-2-en-1-yl)oxy]-5-oxopent-2-enoic acid

651

2934 10 00

136401-69-9

(Z)-5-{4-[2-(5-ethylpyridin-2-yl)ethoxy]benzylidene}-1,3-thiazolidine-2,4-dione

643

2934 10 00

161798-03-4

ethyl 2-(3-formyl-4-isobutoxyphenyl)-4-methylthiazole-5-carboxylate

485

2934 10 00

162208-27-7

O-[2-(2-amino-1,3-thiazol-4-yl)-2-((Z)-methoxyimino)acetyl] O, O-diethyl phosphorothioate

725

2934 10 00

162208-28-8

O-(2-(2-aminothiazol-4-yl)-2-{[1-(tert-butoxycarbonyl)-1-methylethoxy]imino}acetyl) O',O''-diethyl phosphorothioate

46

2934 10 00

179258-52-7

tert-butyl (7Z)-7-(2-amino-1,3-thiazol-5-yl)-4-ethoxy-10,10-dimethyl-6-oxo-3,5,9-trioxa-8-aza-4-phosphaundec-7-en-11-oate 4-oxide

247

2934 10 00

186538-00-1

3-[(2S,3S)-2-hydroxy-3-(3-hydroxy-2-methylbenzamido)-4-phenylbutanoyl]-5,5-dimethyl-N-(2-methylbenzyl)-1,3-thiazolidine-4-carboxamide

104

2934 10 00

189448-35-9

(7R)-7-[(2E)-2-(2-amino-5-chloro-1,3-thiazol-4-yl)-2-(hydroxyimino)acetamido]-3-[(3-{[(2-aminoethyl)sulfanyl]methyl}pyridin-4-yl)sulfanyl]-3,4-didehydrocepham-4-carboxylic acid

388

2934 10 00

213252-19-8

5-[(2,4-dioxo-1,3-thiazolidin-5-yl)methyl]-2-methoxy-N-[4-(trifluoromethyl)benzyl]benzamide

178

2934 10 00

221671-63-2

potassium (2-{N-[4-(4-chloro-2,5-dimethoxyphenyl)-5-(2-cyclohexylethyl)-1,3-thiazol-2-yl]carbamoyl}-5,7-dimethylindolin-1-yl)acetate

111

2934 10 00

224631-15-6

2,5-dioxopyrrolidin-1-yl N-{N-[(2-isopropyl-1,3-thiazol-4-yl)methyl]-N-methylcarbamoyl}-L-valinate

723

2934 10 00

29676-71-9

(2-amino-1,3-thiazol-4-yl)acetic acid

871

2934 10 00

302962-49-8

N-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)thiazole-5-carboxamide or dasatanib (proposed INN)

338

2934 10 00

34272-64-5

(4-methyl-2-sulfanyl-1,3-thiazol-5-yl)acetic acid

859

2934 10 00

478410-84-3

(4R)-N-allyl-3-[(2S,3S)-2-hydroxy-3-(3-hydroxy-2-methylbenzamido)-4-phenylbutanoyl]-5,5-dimethylthiazolidine-4-carboxamide

415

2934 10 00

88023-65-8

potassium 3-[(2-formamido-1,3-thiazol-4-yl)oxoacetamido]-2-methyl-4-oxoazetidine-1-sulfonate

957

2934 99 90

0-00-0

potassium 5-methyl-1,3,4-oxadiazole-2-carboxylate

53

2934 99 90

100988-63-4

1-[((7R)-7-amino-4-carboxy-3,4-didehydrocepham-3-yl)methyl]pyridinium iodide

520

2934 99 90

102212-98-6

N4-benzoyl-2'-deoxy-5'-O-(4,4'-dimethoxytrityl)cytidine 3'-(2-cyanoethyl diisopropylphosphoramidite)

795

2934 99 90

103788-59-6

4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]benzaldehyde

55

2934 99 90

103788-65-4

2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethan-1-ol

618

2934 99 90

110483-43-7

2'-bromo-2'-deoxy-5-methyluridine 3',5'-diacetate

451

2934 99 90

113891-01-3

diphenylmethyl (2S,5R)-6,6-dibromo-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylate 4-oxide

735

2934 99 90

114341-88-7

3-(2-bromopropanoyl)-4,4-dimethyl-1,3-oxazolidin-2-one

343

2934 99 90

127111-98-2

diphenylmethyl (7R)-7-amino-3-(mesyloxy)-3,4-didehydrocepham-4-carboxylate hydrochloride

439

2934 99 90

130800-76-9

5-(3-chloropropyl)-3-methylisoxazole

260

2934 99 90

134379-77-4

4-amino-5-fluoro-1-[(2R,5S)-5-(hydroxymethyl)-2,5-dihydrofuran-2-yl]pyrimidin-2(1H)-one

447

2934 99 90

135790-89-5

[(2,2-dimethylpropanoyl)oxy]methyl (7R)-7-[(2Z)-2-(2-{(2S)-2-[(tert-butoxycarbonyl)amino]propanamido}-1,3-thiazol-4-yl)-2-(methoxyimino)acetamido]-3,4-didehydrocepham-4-carboxylate

767

2934 99 90

13636-02-7

(RS)-3-(dimethylamino)-1-(2-thienyl)propan-1-ol

344

2934 99 90

140128-37-6

diphenylmethyl (7R)-7-(2-{2-[(tert-butoxycarbonyl)amino]-1,3-thiazol-4-yl}-2- [(trityloxy)imino]acetamido)-3-({[(1H-1,2,3-triazol-4-yl)sulfanyl]methyl}sulfanyl)-3,4-didehydrocepham-4-carboxylate

177

2934 99 90

155990-20-8

N-[(1-{[2-(diethylamino)ethyl]amino}-7-methoxy-9-oxo-9H-thioxanthen-4-yl)methyl]formamide

8

2934 99 90

158878-46-7

6-{(E)-2-[4-(4-fluorophenyl)-2,6-diisopropyl-5-(methoxymethyl)pyridin-3-yl]vinyl}-4-hydroxytetrahydro-2H-pyran-2-one

771

2934 99 90

164015-32-1

N-methyl-3-(1-naphthyloxy)-2-(2-thienyl)propan-1-amine phosphate

815A

2934 99 90

170985-86-1

1-[(2S,3S)-2-(benzyloxy)pentan-3-yl]-4-(4-{4-[4-({(3R,5R)-5-(2,4-difluorophenyl)-5-[(1H-1,2,4-triazol-1-yl)methyl]tetrahydrofuran-3-yl}methoxy)phenyl]piperazin-1-yl}phenyl)-1H-1,2,4-triazol-5(4H)-one

382

2934 99 90

171482-05-6

(2R,3S)-2-{(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethoxy}-3-(4-fluorophenyl)morpholine hydrochloride

181

2934 99 90

176773-87-8

(3R)-3-(methoxymethyl)-7-(4,4,4-trifluorobutoxy)-3,3a,4,5-tetrahydro[1,3]oxazolo[3,4-a]quinolin-1-one

278A

2934 99 90

177587-08-5

N-{5-[2-((6S)-2-amino-4-oxo-3,4,5,6,7,8-hexahydropyrido[2,3-d]pyrimidin-6-yl)ethyl]-4-methylthiophene-2-carbonyl}-L-glutamic acid

175

2934 99 90

181640-09-5

3-(1-{2-[4-benzoyl-2-(3,4-difluorophenyl)morpholin-2-yl]ethyl}-4-phenylpiperidin-4-yl)-1,1-dimethylurea hydrochloride

125

2934 99 90

182133-09-1

6-(benzyloxy)-3-bromo-2-(4-methoxyphenyl)-1-benzothiophene 1-oxide

659

2934 99 90

183433-66-1

[6-chloro-4-(2-ethyl-1,3-dioxolan-2-yl)-2-methoxypyridin-3-yl]methanol

242

2934 99 90

183434-04-0

tert-butyl (4S)-4-ethyl-4,6-dihydroxy-3,10-dioxo-3,4,8,10-tetrahydro-1H-pyrano[3,4-f]indolizine-7-carboxylate

182

2934 99 90

185835-97-6

(5S)-5-(methoxymethyl)-3-[6-(4,4,4-trifluorobutoxy)-1,2-benzoxazol-3-yl]-1,3-oxazolidin-2-one

185

2934 99 90

186348-69-6

7-chloro-8-[((2R)-1,4-diazabicyclo[2.2.2]octan-2-yl)methylamino]-2,3-dihydro-1,4-benzodioxine-5-carboxamide

656

2934 99 90

18686-82-3

1,3,4-thiadiazole-2-thiol

252

2934 99 90

188016-51-5

methyl N-(butoxycarbonyl)-3-{[(5R)-3-(4-cyanophenyl)-4,5-dihydroisoxazol-5-yl]acetamido}-L-alaninate

187

2934 99 90

189003-92-7

2-{7-fluoro-2-oxo-4-[2-(4-thieno[3,2-c]pyridin-4-ylpiperazin-1-yl)ethyl]quinolin-1(2H)-yl}acetamide

216

2934 99 90

189028-95-3

(4S)-3-[(5R)-5-(4-fluorophenyl)-5-hydroxypentanoyl]-4-phenyl-1,3-oxazolidin-2-one

186

2934 99 90

191023-43-5

5-(8-amino-7-chloro-2,3-dihydro-1,4-benzodioxin-5-yl)-3-(1-phenethylpiperidin-4-yl)-1,3,4-oxadiazol-2(3H)-one

697

2934 99 90

192049-49-3

4-nitrobenzyl 2-((1R,5R)-3-benzyl-7-oxo-4-thia-2,6-diazabicyclo[3.2.0]hept-2-en-6-yl)-3-methylbut-2-enoate

327

2934 99 90

194861-99-9

((5S)-3-tert-butyl-2-phenyl-1,3-oxazolidin-5-yl)methanol

627

2934 99 90

195708-14-6

(2R,3R,4S)-4-(1,3-benzodioxol-5-yl)-3-(ethoxycarbonyl)-2-(4-methoxyphenyl)pyrrolidinium (2S)-hydroxy(phenyl)acetate

340

2934 99 90

197897-11-3

1-[((7R)-7-amino-4-carboxy-3,4-didehydrocepham-3-yl)methyl]-1H-imidazo[1,2-b]pyridazin-4-ium iodide

30

2934 99 90

199327-61-2

7-methoxy-6-(3-morpholinopropoxy)quinazolin-4(3H)-one

310

2934 99 90

204990-60-3

(3S,10R,13Z,16S)-10-(3-chloro-4-methoxybenzyl)-3-isobutyl-6,6-dimethyl-16-[(1S)-1-((2R,3R)-3-phenyloxiran-2-yl)ethyl]-1,4-dioxa-8,11-diazacyclohexadec-13-ene-2,5,9,12-tetrone

446

2934 99 90

20893-30-5

2-thienylacetonitrile

704B

2934 99 90

220997-99-9

(5R)-9-chloro-5-ethyl-5-hydroxy-10-methyl-12-[(4-methylpiperidin-1-yl)methyl]-1,4,5,13-tetrahydro-3H,15H-oxepino[3',4':6,7]indolizino[1,2-b]quinoline-3,15-dione hydrochloride

704

2934 99 90

221054-70-2

(5R)-5-ethyl-5-hydroxy-1,4,5,8-tetrahydrooxepino[3,4-c]pyridine-3,9-dione

184

2934 99 90

223570-85-2

8-methyl-8-azabicyclo[3.2.1]octan-3-yl 2,3-dihydropyrazolo[1,5,4-de][1,4]benzoxazine-6-carboxylate

432

2934 99 90

223595-20-8

(1R)-5-(1,3,6,2-dioxazaborocan-2-yl)-1-methyl-2-tritylisoindoline

707

2934 99 90

227029-27-8

2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethyl methanesulfonate

299

2934 99 90

227625-35-6

3-{[2-(aminomethyl)cyclohexyl]methyl}-1,2,4-oxadiazol-5(4H)-one

298

2934 99 90

227626-65-5

tert-butyl N-methyl-N-{2-[(5-oxo-4,5-dihydro-1,2,4-oxadiazol-3-yl)methyl]cyclohexyl}carbamate

299A

2934 99 90

227626-75-7

3-{[2-(aminomethyl)cyclohexyl]methyl}-1,2,4-oxadiazol-5(4H)-one hydrochloride

300

2934 99 90

229336-92-9

3-chloro-N-{4-chloro-2-[(5-chloropyridin-2-yl)carbamoyl]-6-methoxyphenyl}-4-{[2-(methylamino)imidazol-1-yl]methyl}thiophene-2-carboxamide

300A

2934 99 90

229340-73-2

3-chloro-N-{4-chloro-2-[(5-chloropyridin-2-yl)carbamoyl]-6-methoxyphenyl}-4-{[2-(methylamino)imidazol-1-yl]methyl}thiophene-2-carboxamide trifluoroacetate

722

2934 99 90

24209-43-6

(7R)-7-amino-3-[2-(1,3,4-thiadiazol-2-ylsulfanyl)ethyl]-3,4-didehydrocepham-4-carboxylic acid

82

2934 99 90

252317-48-9

{(3S)-1-[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl]pyrrolidin-3-yl}diphenylacetonitrile

289

2934 99 90

253450-09-8

6-({2-[4-(4-fluorobenzyl)piperidin-1-yl]ethyl}sulfinyl)-1,3-benzoxazol-2(3H)-one

841

2934 99 90

253450-12-3

6-{[2-(4-benzylpiperidin-1-yl)ethyl]sulfinyl}-1,3-benzoxazol-2(3H)-one

408

2934 99 90

287737-72-8

(2S)-hydroxy(phenyl)acetic acid — (1S)-3-(dimethylamino)-1-(2-thienyl)propan-1-ol (1:1) (salt)

383

2934 99 90

287930-73-8

4-benzyl-2-hydroxymorpholin-3-one

384

2934 99 90

287930-75-0

(2R)-4-benzyl-2-{(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethoxy}morpholin-3-one

325

2934 99 90

30165-96-9

4-(4-chloro-1,2,5-thiadiazol-3-yl)morpholine

815

2934 99 90

345217-03-0

2-[(2S,3S)-2-(benzyloxy)pentan-3-yl]-4-(4-{4-[4-({(3R,5R)-5-(2,4-difluorophenyl)-5-[(1H-1,2,4-triazol-1-yl)methyl]tetrahydrofuran-3-yl}methoxy)phenyl]piperazin-1-yl}phenyl)semicarbazide

854

2934 99 90

362543-73-5

DNA, d(P-thio) (C-T-A-G-A-T-T-T-C-C-C-G-C-G), tridecasodium salt

448

2934 99 90

36923-17-8

(7R)-7-amino-3,4-didehydrocepham-4-carboxylic acid

717

2934 99 90

37539-03-0

(7R)-7-amino-3-[(1H-1,2,3-triazol-4-ylsulfanyl)methyl]-3,4-didehydrocepham-4-carboxylic acid

832

2934 99 90

377727-87-2

2-(2-furyl)-7-(2-{4-[4-(2-methoxyethoxy)phenyl]piperazin-1-yl}ethyl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[2,3-c]pyrimidin-5-amine

706B

2934 99 90

475479-34-6

(2S)-2-methoxy-3-{4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]-1-benzothiophen-7-yl}propanoic acid

706

2934 99 90

475480-88-7

4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]-1-benzothiophene-7-carbaldehyde

959

2934 99 90

518048-05-0

potassium 4-[N-(2-fluorobenzyl)carbamoyl]-1-methyl-2-[1-methyl-1-(5-methyl-1,3,4-oxadiazole-2-carboxamido)ethyl]-6-oxo-1,6-dihydropyrimidine-5-olate

707A

2934 99 90

521266-46-6

(2S)-1-{N-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethyl]glycyl}pyrrolidine-2-carbonitrile

655

2934 99 90

53994-69-7

(7R)-7-amino-3-chloro-3,4-didehydrocepham-4-carboxylic acid

719

2934 99 90

61807-78-1

7-(bromoacetamido)-7-methoxy-3-{[(1-methyl-1H-tetrazol-5-yl)lsulfanyl]methyl}-3,4-didehydrocepham-4-carboxylic acid

738

2934 99 90

63457-21-6

diphenylmethyl 2-(3-benzyl-7-oxo-4-thia-2,6-diazabicyclo[3.2.0]hept-2-en-6-yl)-3-methylbut-3-enoate

961

2934 99 90

635724-55-9

(2S)-2-[(S)-(2-ethoxyphenoxy)phenylmethyl]morpholine succinate

797

2934 99 90

649761-25-1

methyl N-{4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]benzyl}glycinate hydrochloride

702

2934 99 90

655233-39-9

4-nitrobenzyl (7R)-7-amino-3-((2S)-tetrahydrofuran-2-yl)-3,4-didehydrocepham-4-carboxylate hydrochloride

769

2934 99 90

663603-70-1

(2Z)-3-(methylamino)-1-(2-thienyl)prop-2-en-1-one

721

2934 99 90

68350-02-7

(7R)-7-amino-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}-3,4-didehydrocepham-4-carboxylic acid hydrochloride

718

2934 99 90

70035-75-5

diphenylmethyl (7S)-7-(bromoacetamido)-7-methoxy-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}-3,4-didehydrocepham-4-carboxylate

855

2934 99 90

744239-10-9

DNA, d(P-thio) (G-A-T-C-C-G-C-G-G-G-A-A-A-T), tridecasodium salt

665

2934 99 90

7481-90-5

1-(3,5-anhydro-2-deoxy-β-D-threo-pentofuranosyl)-5-methylpyrimidine-2,4(1H,3H)-dione

208

2934 99 90

75776-79-3

1,4-dithia-7-azaspiro[4.4]nonane-8-carboxylic acid hydrobromide

93

2934 99 90

76646-91-8

(3S)-6,6-dibromo-2,2-dimethylpenam-3-carboxylic acid 1,1-dioxide

90

2934 99 90

76801-85-9

(2R,3S,4R,5R,8R,10R,11R,12S,13S,14R)-13-[(2,6-dideoxy-3-C-methyl-3-O-methyl-α-L-ribo-hexopyranosyl)oxy]-2-ethyl-3,4,10-trihydroxy-3,5,8,10,12,14-hexamethyl-11-{[3,4,6-trideoxy-3-(dimethylamino)-β-D-xylo-hexopyranosyl]oxy}-1-oxa-6-azacyclopentadecan-15-one

716

2934 99 90

79349-82-9

trans-(7R)-7-amino-3-vinyl-3,4-didehydrocepham-4-carboxylic acid

243

2934 99 90

86639-52-3

(4S)-4,11-diethyl-4,9-dihydroxy-1H,12H-pyrano[3',4':6,7]indolizino[1,2-b]quinoline-3,14(4H,12H)-dione

952

2934 99 90

872728-82-0

N-[4-(5-oxo-4,5-dihydro-1,2,4-oxadiazol-3-yl)phenyl]glycine

342

2934 99 90

92096-37-2

diphenylmethyl (7R)-3-(mesyloxy)-7-(phenylacetamido)-3,4-didehydrocepham-4-carboxylate

525

2934 99 90

93183-15-4

2'-deoxy-5'-O-(4,4'-dimethoxytrityl)-N2-isobutyrylguanosine 3'-(2-cyanoethyl diisopropylphosphoramidite)

688

2934 99 90

96219-87-3

(3-aminopyrazol-4-yl)(2-thienyl)methanone

584

2934 99 90

98-03-3

thiophene-2-carbaldehyde

526

2934 99 90

98796-51-1

2'-deoxy-5'-O-(4,4'-dimethoxytrityl)thymidine 3'-(2-cyanoethyl diisopropylphosphoramidite)

527

2934 99 90

98796-53-3

N6-benzoyl-2'-deoxy-5'-O-(4,4'-dimethoxytrityl)adenosine 3'-(2-cyanoethyl diisopropylphosphoramidite)

517

2934 99 90

98819-76-2

(2S)-2-[(S)-(2-ethoxyphenoxy)phenylmethyl]morpholine

770

2934 99 90

116539-55-0

(1S)-3-(methylamino)-1-(2-thienyl)propan-1-ol

179

2935 00 90

137431-02-8

N-[3-(2-amino-1-hydroxyethyl)-4-fluorophenyl]methanesulfonamide

626a

2935 00 90

141430-65-1

N-[2-(4-hydroxyanilino)pyridin-3-yl]-4-methoxybenzene-1-sulfonamide

329

2935 00 90

149490-60-8

N-(butane-1-sulfonyl)-L-tyrosine

328

2935 00 90

149490-61-9

N-(butane-1-sulfonyl)-O-(4-pyridin-4-ylbutyl)-L-tyrosine

40

2935 00 90

160231-69-6

(3S)-tetrahydrofuran-3-yl N-[(2S,3R)-3-hydroxy-4-(N-isobutyl-4-nitrobenzene-1-sulfonamido)-1-phenylbutan-2-yl]carbamate

562

2935 00 90

169280-56-2

4-amino-N-[(2R,3S)-3-amino-2-hydroxy-4-phenylbutyl]-N-isobutylbenzene-1-sulfonamide

711

2935 00 90

170569-88-7

4-[5-(4-fluorophenyl)-3-(trifluoromethyl)pyrazol-1-yl]benzene-1-sulfonamide

691

2935 00 90

186497-07-4

N-(3-methoxy-5-methylpyrazin-2-yl)-2-[4-(1,3,4-oxadiazol-2-yl)phenyl]pyridine-3-sulfonamide

180

2935 00 90

189814-01-5

3-(2-amino-1-hydroxyethyl)-4-methoxybenzene-1-sulfonamide

88

2935 00 90

200575-15-1

4-[2-ethoxy-5-(4-methylpiperazine-1-sulfonyl)benzamido]-1-methyl-3-propylpyrazole-5-carboxamide

587

2935 00 90

210538-75-3

N-(1,2,3,4-tetrahydroisoquinolin-5-yl)methanesulfonamide hydrochloride

41

2935 00 90

244634-31-9

N-((2R,3S)-3-amino-2-hydroxy-4-phenylbutyl)-N-isobutyl-4-nitrobenzene-1-sulfonamide hydrochloride

75

2935 00 90

247582-73-6

2-ethoxy-5-(4-ethylpiperazine-1-sulfonyl]nicotinic acid

224

2935 00 90

289042-12-2

(4R,6S)-6-((E)-2-{4-(4-fluorophenyl)-6-isopropyl-2-[mesyl(methyl)amino]pyrimidin-5-yl}vinyl)-2,2-dimethyl-1,3-dioxan-4-yl 3,3-dimethylbutanoate

592

2935 00 90

334826-98-1

5-[2-ethoxy-5-(4-ethylpiperazine-1-sulfonyl)pyridin-3-yl]-3-ethyl-2-(2-methoxyethyl)-2,3,4,5,6,7-hexahydropyrazolo[4,3-d]pyrimidin-7-one

593

2935 00 90

334827-99-5

5-[2-ethoxy-5-(4-ethylpiperazine-1-sulfonyl)pyridin-3-yl]-3-ethyl-2-(2-methoxyethyl)-2,3,4,5,6,7-hexahydropyrazolo[4,3-d]pyrimidin-7-one 4-methylbenzene-1-sulfonate

591

2935 00 90

334828-19-2

N-[3-carbamoyl-5-ethyl-1-(2-methoxyethyl)pyrazol-4-yl]-2-ethoxy-5-[(4-ethylpiperazin-1-yl)sulfonyl]nicotinamide

596

2935 00 90

364321-71-1

3-[(dimethylamino)methyl]-4-[4-(methylsulfanyl)phenoxy]benzene-1-sulfonamide

597

2935 00 90

364323-49-9

3-[(dimethylamino)methyl]-4-[4-(methylsulfanyl)phenoxy]benzene-1-sulfonamide L-tartarate (1:1)

70

2935 00 90

88933-16-8

1-(4-hydrazinophenyl)-N-methylmethanesulfonamide hydrochloride

335

2938 90 90

517-43-1

mixture of sennoside A and B

336

2938 90 90

52730-36-6 , 52730-37-7

mixture of sennoside A and B, calcium salts

882

2939 19 00

58-00-4

(6aR)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de, g]quinoline-10,11-diol or apomorphine

666

2939 20 00

467430-13-3

2-[2-methyl-1-(propionyloxy)propoxy]-2-[(4-phenylbutyl)phosphinoyl]acetic acid, (9R)-cinchonan-9-ol salt (1:1)

617

2940 00 00

270071-40-4

benzyl 2,6-dimethoxy-4-{(5R,5aR,8aR,9S)-6-oxo-9-[(2,3,4,6-tetra-O-benzyl-β-D-glucopyranosyl)oxy]-5,5a,6,8,8a,9-hexahydrofuro[3',4':6,7]naphtho[2,3-d][1,3]dioxol-5-yl}phenyl carbonate

667

2940 00 00

471863-88-4

2,3-di-O-benzyl-4,6-O-((1R)-ethylidene)-D-xylo-hexopyranose

668

2940 00 00

473799-30-3

(5S,5aS,9S)-9-(4-hydroxy-3,5-dimethoxyphenyl)-8-oxo-5,5a,6,8,8a,9-hexahydrofuro[3',4':6,7]naphtho[2,3-d][1,3]dioxol-5-yl 2,3-di-O-benzyl-4,6-O-[(1R)-ethylidene]-β-D-glucopyranoside

616

2940 00 00

6564-72-3

2,3,4,6-tetra-O-benzyl-D-glucopyranose

15

2941 90 00

19130-96-2

(2S,3S,4R,5R)-2-(hydroxymethyl)piperidine-3,4,5-triol

200

2941 90 00

54122-50-8

dicyclohexylammmonium (7R)-3-(acetoxymethyl)-7-[2-({(3R)-3-[(tert-butoxycarbonyl)amino]-3-carboxypropyl}amino)-2-oxoethyl]-3,4-didehydrocepham-4-carboxylate or cephalosporin D dicyclohexylamine salt

131

3002 10 95

42617-41-4

Blood-coagulation factor XIVa

321

3824 90 98

127852-28-2

(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethan-1-ol, acetonitrile solution

510

3824 90 98

170277-77-7

(3S)-3-[2-(mesyloxy)ethoxy]-4-(trityloxy)butyl methanesulfonate, dimethylformamide solution

326

3824 90 98

30165-96-9

4-(4-chloro-1,2,5-thiadiazol-3-yl)morpholine, toluene solution

409

3824 90 98

38345-66-3

(2S,3R)-4-(dimethylamino)-3-methyl-1,2-diphenylbutan-2-ol, toluene solution

132

3824 90 98

84449-81-0

4-[2-(piperidin-1-yl)ethoxy]benzoyl chloride hydrochloride, 1,2-dichloroethane solution

ANNEX IV

List of pharmaceutical intermediates, i.e. compounds used for the manufacture of finished pharmaceutical products, to be withdrawn from the list of products receiving duty-free treatment included in Annex 6 to Regulation (EC) No 1549/2006

ID No

CN code

CAS RN

Name

677

2918 90 90

157283-68-6

isopropyl (Z)-7-[(1R,2R,3R,5S)-3,5-dihydroxy-2-{(E)-(3R)-3-hydroxy-4-[3-(trifluoromethyl)phenoxy]but-1-enyl}cyclopentyl]hept-5-enoate

travoprost (INN)

603

2924 29 95

112522-64-2

4-acetamido-2'-aminobenzanilide

tacedinaline (INN)

69

2924 29 95

166518-60-1

N-[(2,6-diisopropylphenoxy)sulfonyl]-2-(2,4,6-triisopropylphenyl)acetamide

avasimibe (INN)

441

2928 00 90

53016-31-2

13-ethyl-17-alpha-hydroxy-18,19-dinorpregn-4-en-20-yn-3-one oxime

norelgestromin (INN)

833

2930 90 30

583-91-5

2-hydroxy-4-(methylthio)butyric acid

desmeninol (INN)

273

2932 99 70

114870-03-0

methyl O-2-deoxy-6-O-sulfo-2-(sulfoamino)-alpha-D-glucopyranosyl-(1,4)-O-beta-D-glucopyranuronosyl-(1,4)-O-2-deoxy-3,6-di-O-sulfo-2-(sulfoamino)-alpha-D-glucopyranosyl-(1,4)-O-2-O-sulfo-alpha-L-idopyranuronosyl-(1,4)-2-deoxy-2-(sulfoamino)-6-(hydrogen sulfate)-alpha-D-glucopyranoside, decasodium salt

fondaparinux sodium (INN)

627

2933 39 99

75970-99-9

[1-(4-fluorobenzyl)-1H-benzimidazol-2-yl](4-piperidyl)amine

tecastemizole (INN)

159

2933 39 99

100643-71-8

8-chloro-11-(4-piperidylidene)-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridine

desloratadine (INN)

549

2933 39 99

168273-06-1

5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-piperidino-1H-pyrazole-3-carboxamide

rimonabant (INN)

380

2933 39 99

193275-84-2

4-{4-[(11R)-3,10-dibromo-8-chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-yl]piperidinocarbonylmethyl}piperidine-1-carboxamide

lonafarnib (INN)

397

2933 49 90

146362-70-1

2-{[1-(7-chloro-4-quinolyl)-5-(2,6-dimethoxyphenyl)-1H-pyrazol-3-yl]carbonylamino}adamantane-2-carboxylic acid

meclinertant (INN)

641

2933 59 95

147127-20-6

(R)-[2-(6-amino-9H-purin-9-yl)-1-methylethoxy]methylphosphonic acid

tenofovir (INN)

205

2933 59 95

149950-60-7

6-benzyl-1-(ethoxymethyl)-5-isopropylpyrimidine-2,4(1H,3H)-dione

emivirine (INN)

511

2933 59 95

153537-73-6

(S)-2-(4-{[(2,7-dimethyl-4-oxo-1,4-dihydroquinazolin-6-yl)methyl](prop-2-ynyl)amino}-2-fluorobenzamido)-4-(1H-tetrazol-5-yl)butyric acid

plevitrexed (INN)

686

2934 99 90

112984-60-8

(+-)-6-fluoro-1-methyl-4-oxo-7-(piperazin-1-yl)-4H-[1,3]thiazeto[3,2-a]quinoline-3-carboxylic acid

ulifloxacin (INN)

33

2934 99 90

145514-04-1

(2R,4R)-4-(2,6-diamino-9H-purin-9-yl)-1,3-dioxolan-2-ylmethanol

amdoxovir (INN)

513

2934 99 90

171228-49-2

4-[4-(4-{4-[(3R,5R)-5-(2,4-difluorophenyl)-5-(1H-1,2,4-triazol-1-ylmethyl)tetrahydrofuran-3-ylmethyloxy]phenyl}piperazin-1-yl)phenyl]-1-[(1S,2S)-1-ethyl-2-hydroxypropyl]-1,2,4-triazol-5(4H)-one

posaconazole (INN)

293

2934 99 90

184475-35-2

(3-chloro-4-fluorophenyl)[7-methoxy-6-(3-morpholinopropoxy)quinazolin-4-yl]amine

gefitinib (INN)

539

2935 00 90

150375-75-0

N'-{(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-3-hydroxy-2,3-dihydro-1H-indol-2-ylcarbonyl}-L-prolinamide

relcovaptan (INN)

39

2935 00 90

161814-49-9

(3S)-tetrahydrofuran-3-yl (1S,2R)-3-[(4-aminophenylsulfonyl)(isobutyl)amino]-1-benzyl-2-hydroxypropylcarbamate

amprenavir (INN)

115

2935 00 90

169590-42-5

4-[5-(p-tolyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl]benzenesulfonamide

celecoxib (INN)

654

2935 00 90

180200-68-4

4-(4-cyclohexyl-2-methyloxazol-5-yl)-2-fluorobenzenesulfonamide

tilmacoxib (INN)

690

2935 00 90

181695-72-7

4-(5-methyl-3-phenylisoxazol-4-yl)benzenesulfonamide

valdecoxib (INN)

520

2935 00 90

192329-42-3

(S)-N-hydroxy-2,2-dimethyl-4-[4-(4-pyridyloxy)phenylsulfonyl]-1,4-thiazinane-3-carboxamide

prinomastat (INN)

364

3002 10 95

193700-51-5

SC-70935

leridistim (INN)

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